An intracellular targeted antibody detects EGFR as an independent prognostic factor in ovarian carcinomas

BMC Cancer. 2011 Jul 14:11:294. doi: 10.1186/1471-2407-11-294.

Abstract

Background: In ovarian cancer, the reported rate of EGFR expression varies between 4-70% depending on assessment method and data on patient outcome are conflicting.

Methods: In this study we investigated EGFR expression and its prognostic value in a cohort of 121 invasive ovarian carcinomas, using a novel antibody against the intracellular domain of the receptor. We further evaluated an association between EGFR, the nuclear transporter CRM1 as well as COX-2. Furthermore, we evaluated EGFR expression in ten ovarian cancer cell lines and incubated cancer cells with Leptomycin B, a CRM1 specific inhibitor.

Results: We observed a membranous and cytoplasmic EGFR expression in 36.4% and 64% of ovarian carcinomas, respectively. Membranous EGFR was an independent prognostic factor for poor overall survival in ovarian cancer patients (HR 2.7, CI 1.1-6.4, p = 0.02) which was also found in the serous subtype (HR 4.6, CI 1.6-13.4, p = 0.004). We further observed a significant association of EGFR with COX-2 and nuclear CRM1 expression (chi-square test for trends, p = 0.006 and p = 0.013, respectively). In addition, combined membranous EGFR/COX-2 expression was significantly related to unfavorable overall survival (HR 7.2, CI 2.3-22.1, p = 0.001).In cell culture, we observed a suppression of EGFR protein levels after exposure to Leptomycin B in OVCAR-3 and SKOV-3 cells.

Conclusions: Our results suggest that the EGFR/COX-2/CRM1 interaction might be involved in progression of ovarian cancer and patient prognosis. Hence, it is an interesting anti-cancer target for a combination therapy. Further studies will also be needed to investigate whether EGFR is also predictive for benefit from EGFR targeted therapies.

MeSH terms

  • Adult
  • Aged
  • Aged, 80 and over
  • Animals
  • Antibodies, Monoclonal / immunology*
  • Antibodies, Neoplasm / immunology*
  • Antibody Specificity
  • Biomarkers, Tumor / analysis*
  • Biomarkers, Tumor / immunology
  • Carcinoma / chemistry*
  • Carcinoma / mortality
  • Carcinoma / pathology
  • Cell Line, Tumor / drug effects
  • Cell Line, Tumor / metabolism
  • Cohort Studies
  • Cyclooxygenase 2 / analysis
  • ErbB Receptors / analysis*
  • ErbB Receptors / biosynthesis
  • ErbB Receptors / genetics
  • ErbB Receptors / immunology
  • Exportin 1 Protein
  • Fatty Acids, Unsaturated / pharmacology
  • Female
  • Gene Expression Regulation, Neoplastic / drug effects
  • Humans
  • Immunoenzyme Techniques
  • Kaplan-Meier Estimate
  • Karyopherins / analysis
  • Karyopherins / antagonists & inhibitors
  • Middle Aged
  • Neoplasm Proteins / analysis*
  • Neoplasm Proteins / antagonists & inhibitors
  • Neoplasm Proteins / biosynthesis
  • Neoplasm Proteins / genetics
  • Neoplasm Proteins / immunology
  • Ovarian Neoplasms / chemistry*
  • Ovarian Neoplasms / mortality
  • Ovarian Neoplasms / pathology
  • Prognosis
  • Protein Structure, Tertiary
  • Rabbits
  • Receptors, Cytoplasmic and Nuclear / analysis
  • Receptors, Cytoplasmic and Nuclear / antagonists & inhibitors
  • Single-Blind Method

Substances

  • Antibodies, Monoclonal
  • Antibodies, Neoplasm
  • Biomarkers, Tumor
  • Fatty Acids, Unsaturated
  • Karyopherins
  • Neoplasm Proteins
  • Receptors, Cytoplasmic and Nuclear
  • Cyclooxygenase 2
  • PTGS2 protein, human
  • EGFR protein, human
  • ErbB Receptors
  • leptomycin B