[Effects of glycyrrhiza extract on pharmacokinetics property of daphnetin in rats]

Zhongguo Zhong Yao Za Zhi. 2011 Apr;36(7):935-8.
[Article in Chinese]

Abstract

Objective: To research the influence of glycyrrhiza extract on the pharmacokinetics characteristic parameters of daphnetin, which was aimed to explore the rationality of concert application of drugs.

Method: The rats received intragastric administration of daphnetin and glycyrrhiza extract containing the same daphnetin respectively. The blood concentration of daphnetin was assayed by LC-MS. The data was processed by program DAS2.1.1.

Result: Glycyrrhiza extract can reduce the t(1/2), tmax and Ke of daphnetin, while increased the Ka and AUC(0-infinity).

Conclusion: Glycyrrhiza extract promoted the oral absorption of daphnetin, slowed down the elimination and increased the biological availability.

Publication types

  • English Abstract

MeSH terms

  • Animals
  • Drug Interactions
  • Drugs, Chinese Herbal / pharmacology*
  • Glycyrrhiza / chemistry*
  • Rats
  • Rats, Sprague-Dawley
  • Tissue Distribution / drug effects
  • Umbelliferones / pharmacokinetics*

Substances

  • Drugs, Chinese Herbal
  • Umbelliferones
  • daphnetin