Appropriateness and complications of the use of spironolactone in patients treated in a heart failure clinic

Eur J Intern Med. 2011 Aug;22(4):424-7. doi: 10.1016/j.ejim.2011.04.008. Epub 2011 May 31.

Abstract

Objectives: The widespread use of spironolactone in patients with congestive heart failure (CHF) has resulted in side effects and complications. We analyzed a cohort of patients treated by a dedicated CHF team, in order to examine the tolerability and safety of spironolactone in clinical practice.

Methods: We retrospectively evaluated data on 157 patients who were followed by the Heart Failure clinic of whom 100 patients on maximal treatment (all on β blockers, 99% on ACE inhibitors) received spironolactone. The complications following spironolactone use were defined as: hyperkalemia with serum K 5.2 mEq/l; creatinine 2.0 mg/dl; hyponatremia with serum Na 135 mEq/l, hypotension and side effects such as gynecomastia and abdominal pain.

Results: At 1 year follow-up 6 patients developed hyperkalemia (range 5.3-5.9), 4 of them had K>5.5 mEq/l. Two patients developed hyponatremia. Six patients stopped spironolactone for: 1-gynecomastia, 2-worsening renal failure and hyperkalemia, 2-hyperkalemia (5.9 mEq/l) and 1 for bradycardia. There was an increase in mean creatinine level at 1 year (1.12±0.35 vs. 1.21±0.38 mg/dl, p=0.02), however, no significant changes were found in GFR (99.9±33.5 vs. 65.7±27.7 ml min(-1)1.73 m(-2), p=ns) and potassium (4.5±0.4 vs. 4.6±0.5 mEq/l, p=ns). We found improvement of GFR by >10% in 19 patients and worsening by >10% in 38 patients. No patient was hospitalized or required urgent treatment for spironolactone-related side effects.

Conclusions: In patients with CHF on optimal therapy with ACE inhibitors and β blockers appropriate spironolactone use and close follow-up by a dedicated HF team can minimize the risk for adverse events and complications.

Publication types

  • Comparative Study

MeSH terms

  • Aged
  • Diuretics / administration & dosage
  • Diuretics / adverse effects
  • Diuretics / therapeutic use*
  • Dose-Response Relationship, Drug
  • Female
  • Follow-Up Studies
  • Heart Failure / drug therapy*
  • Hospitals, Special*
  • Humans
  • Hyperkalemia / chemically induced*
  • Male
  • Mineralocorticoid Receptor Antagonists / administration & dosage
  • Retrospective Studies
  • Spironolactone / administration & dosage
  • Spironolactone / adverse effects
  • Spironolactone / therapeutic use*
  • Time Factors
  • Treatment Outcome

Substances

  • Diuretics
  • Mineralocorticoid Receptor Antagonists
  • Spironolactone