Binding characteristics of thrombin-activatable fibrinolysis inhibitor to streptococcal surface collagen-like proteins A and B

Thromb Haemost. 2011 Oct;106(4):609-16. doi: 10.1160/TH11-03-0204. Epub 2011 Jul 28.

Abstract

Streptococcus pyogenes is the causative agent in a wide range of diseases in humans. Thrombin-activatable fibrinolysis inhibitor (TAFI) binds to collagen-like proteins SclA and SclB at the surface of S. pyogenes. Activation of TAFI at this surface redirects inflammation from a transient to chronic state by modulation of the kallikrein/kinin system. We investigated TAFI binding characteristics to SclA/SclB. Thirty-four overlapping TAFI peptides of ~20 amino acids were generated. Two of these peptides (P18: residues G205-S221, and P19: R214-D232) specifically bound to SclA/SclB with high affinity, and competed in a dose-dependent manner with TAFI binding to SclA/SclB. In another series of experiments, the binding properties of activated TAFI (TAFIa) to SclA/SclB were studied with a quadruple TAFI mutant (TAFI-IIYQ) that after activation is a 70-fold more stable enzyme than wild-type TAFIa. TAFI and TAFI-IIYQ bound to the bacterial proteins with similar affinities. The rate of dissociation was different between the proenzyme (both TAFI and TAFI-IIYQ) and the stable enzyme TAFIa-IIYQ. TAFIa-IIYQ bound to SclA/SclB, but dissociated faster than TAFI-IIYQ. In conclusion, the bacterial proteins SclA and SclB bind to a TAFI fragment encompassing residues G205-D232. Binding of TAFI to the bacteria may allow activation of TAFI, whereafter the enzyme easily dissociates.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Sequence
  • Bacterial Proteins / chemistry
  • Bacterial Proteins / metabolism
  • Blood Coagulation Disorders / blood*
  • Blood Coagulation Disorders / etiology
  • Blood Coagulation Disorders / microbiology
  • Carboxypeptidase B2 / chemistry*
  • Carboxypeptidase B2 / genetics
  • Carboxypeptidase B2 / metabolism
  • Enzyme Activation
  • Exotoxins / chemistry
  • Exotoxins / metabolism
  • Humans
  • Membrane Proteins / chemistry
  • Membrane Proteins / metabolism
  • Molecular Sequence Data
  • Mutation / genetics
  • Peptide Fragments / chemistry*
  • Peptide Fragments / genetics
  • Peptide Fragments / metabolism
  • Protein Binding
  • Protein Stability
  • Streptococcal Infections / blood*
  • Streptococcal Infections / complications
  • Streptococcal Infections / microbiology
  • Streptococcus pyogenes / metabolism
  • Streptococcus pyogenes / pathogenicity*
  • Thrombin / metabolism

Substances

  • Bacterial Proteins
  • Exotoxins
  • Membrane Proteins
  • Peptide Fragments
  • SpeA protein, Streptococcus pyogenes
  • erythrogenic toxin
  • Carboxypeptidase B2
  • Thrombin