Self-catalyzed degradable cationic polymer for release of DNA

Biomacromolecules. 2011 Oct 10;12(10):3540-8. doi: 10.1021/bm2007423. Epub 2011 Aug 31.

Abstract

The controlled release of siRNA or DNA complexes from cationic polymers is an important parameter design in polymer-based delivery carriers. In this work, we use the self-catalyzed degradable poly(2-dimethylaminoethyl acrylate) (PDMAEA) to strongly bind, protect, and then release oligo DNA (a mimic for siRNA) without the need for a cellular or external trigger. This self-catalyzed hydrolysis process of PDMAEA forms poly(acrylic acid) and N,N'-dimethylamino ethyl ethanol, both of which have little or no toxicity to cells, and offers the advantage of little or no toxicity to off-target cells and tissues. We found that PDMAEA makes an ideal component of a delivery carrier by protecting the oligo DNA for a sufficiently long period of time to transfect most cells (80% transfection after 4 h) and then has the capacity to release the DNA inside the cells after ~10 h. The PDMAEA formed large nanoparticle complexes with oligo DNA of ~400 nm that protected the oligo DNA from DNase in serum. The nanoparticle complexes showed no toxicity for all molecular weights at a nitrogen/phosphorus (N/P) ratio of 10. Only the higher molecular weight polymers at very high N/P ratios of 200 showed significant levels of cytotoxicity. These attributes make PDMAEA a promising candidate as a component in the design of a gene delivery carrier without the concern about accumulated toxicity of nanoparticles in the human body after multiadministration, an issue that has become increasingly more important.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Acrylic Resins / chemistry*
  • Biocompatible Materials / chemistry*
  • Biocompatible Materials / metabolism
  • Biocompatible Materials / pharmacology
  • Catalysis
  • Cations / chemistry
  • Cations / metabolism
  • Cell Survival / drug effects
  • Delayed-Action Preparations / chemistry*
  • Delayed-Action Preparations / metabolism
  • Delayed-Action Preparations / pharmacology
  • Female
  • Gene Transfer Techniques*
  • HeLa Cells
  • Humans
  • Hydrogen-Ion Concentration
  • Hydrolysis
  • Kinetics
  • Molecular Mimicry
  • Nanoparticles
  • Oligodeoxyribonucleotides / metabolism*
  • Oligodeoxyribonucleotides / pharmacology
  • Particle Size
  • RNA, Small Interfering / metabolism
  • RNA, Small Interfering / pharmacology
  • Spectrometry, Mass, Matrix-Assisted Laser Desorption-Ionization

Substances

  • Acrylic Resins
  • Biocompatible Materials
  • Cations
  • Delayed-Action Preparations
  • Oligodeoxyribonucleotides
  • RNA, Small Interfering
  • carbopol 940