Cell cycle-regulated multi-site phosphorylation of Neurogenin 2 coordinates cell cycling with differentiation during neurogenesis

Development. 2011 Oct;138(19):4267-77. doi: 10.1242/dev.067900. Epub 2011 Aug 18.

Abstract

During development of the central nervous system, the transition from progenitor maintenance to differentiation is directly triggered by a lengthening of the cell cycle that occurs as development progresses. However, the mechanistic basis of this regulation is unknown. The proneural transcription factor Neurogenin 2 (Ngn2) acts as a master regulator of neuronal differentiation. Here, we demonstrate that Ngn2 is phosphorylated on multiple serine-proline sites in response to rising cyclin-dependent kinase (cdk) levels. This multi-site phosphorylation results in quantitative inhibition of the ability of Ngn2 to induce neurogenesis in vivo and in vitro. Mechanistically, multi-site phosphorylation inhibits binding of Ngn2 to E box DNA, and inhibition of DNA binding depends on the number of phosphorylation sites available, quantitatively controlling promoter occupancy in a rheostat-like manner. Neuronal differentiation driven by a mutant of Ngn2 that cannot be phosphorylated by cdks is no longer inhibited by elevated cdk kinase levels. Additionally, phosphomutant Ngn2-driven neuronal differentiation shows a reduced requirement for the presence of cdk inhibitors. From these results, we propose a model whereby multi-site cdk-dependent phosphorylation of Ngn2 interprets cdk levels to control neuronal differentiation in response to cell cycle lengthening during development.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Basic Helix-Loop-Helix Transcription Factors / metabolism*
  • Cell Cycle
  • Cell Differentiation
  • Gene Expression Regulation, Developmental*
  • HeLa Cells
  • Humans
  • Mice
  • Models, Biological
  • Mutation
  • Nerve Tissue Proteins / metabolism*
  • Neurogenesis*
  • Neurons / cytology
  • Phosphorylation
  • Xenopus Proteins / metabolism*
  • Xenopus laevis

Substances

  • Basic Helix-Loop-Helix Transcription Factors
  • NEUROG2 protein, Xenopus
  • Nerve Tissue Proteins
  • Neurog2 protein, mouse
  • Xenopus Proteins