Induction of heme oxygenase 1 prevents progression of liver fibrosis in Mdr2 knockout mice

Hepatology. 2012 Feb;55(2):553-62. doi: 10.1002/hep.24711.

Abstract

Induction or overexpression of the heme-degrading enzyme, heme oxygenase 1 (HO-1), has been shown to protect mice from liver damage induced by acute inflammation. We have investigated the effects of HO-1 induction in a mouse model of chronic liver inflammation and fibrogenesis with progression to hepatocellular carcinoma (HCC) (Mdr2ko; FVB.129P2-Abcb4(tm1Bor)). HO-1 was induced in vivo by treatment with cobalt protoporphyrin IX, starting at week 5 or 12 of mice lifespan, and continued for 7 weeks. Our results showed that HO-1 induction reduced liver damage and chronic inflammation by regulating immune cell infiltration or proliferation as well as tumor necrosis factor receptor signaling. Fibrosis progression was significantly reduced by HO-1 induction in mice with mild, as well as established, portal and lobular fibrosis. HO-1 induction significantly suppressed hepatic stellate cell activation. During established fibrosis, HO-1 induction was able to revert portal inflammation and fibrosis below levels observed at the start of treatment. Moreover, hepatocellular proliferation and signs of dysplasia were decreased after HO-1 induction.

Conclusion: Induction of HO-1 interferes with chronic inflammation and fibrogenesis and, in consequence, might delay progression to HCC.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • ATP Binding Cassette Transporter, Subfamily B / genetics
  • ATP-Binding Cassette Sub-Family B Member 4
  • Animals
  • Cell Proliferation
  • Disease Progression
  • Extracellular Signal-Regulated MAP Kinases / metabolism
  • Female
  • Heme Oxygenase-1 / metabolism*
  • Liver Cirrhosis / enzymology*
  • Liver Cirrhosis / immunology
  • Membrane Proteins / metabolism*
  • Mice
  • Mice, Knockout
  • Phosphorylation
  • Protoporphyrins
  • Receptors, Tumor Necrosis Factor / metabolism

Substances

  • ATP Binding Cassette Transporter, Subfamily B
  • Membrane Proteins
  • Protoporphyrins
  • Receptors, Tumor Necrosis Factor
  • cobaltiprotoporphyrin
  • Heme Oxygenase-1
  • Hmox1 protein, mouse
  • Extracellular Signal-Regulated MAP Kinases