Isolation of two high-molecular-mass proteinases from human erythrocytes

Eur J Biochem. 1990 Jul 31;191(2):275-80. doi: 10.1111/j.1432-1033.1990.tb19120.x.

Abstract

Two forms of a neutral--alkaline high-molecular-mass proteinase (termed A1 and A2) have been purified from human erythrocytes by a procedure including a DEAE-cellulose batchwise treatment of erythrocyte cytosol, gel filtration and DEAE-cellulose chromatography. Both enzymes show distinctive properties of multicatalytic proteinases. They have an apparent molecular mass of 700 kDa and are composed by eight major subunits (23-32 kDa). Both enzymes show a proteinase activity towards casein and hydrolyze synthetic peptides with tyrosine, arginine or lysine at the P1 position. Among the synthetic peptides tested, the tetrapeptide succinyl-leucyl-leucyl-valyl-tyrosyl-7-amido-4-methylcoumarin and tripeptides with arginine in the P1 position (benzyloxycarbonyl-valyl-leucyl-arginyl-4-methoxy-2-naphthylamide and benzyloxycarbonyl-alanyl-arginyl-arginyl-4-methoxy-2-naphthylamide) are the most effective substrates. The proteinases are devoid of amino and diaminopeptidase activity. Both enzymes are completely inhibited by hemin, chymostatin and thiol-group reagents. However, the enzymes can be distinguished by the isoelectric point, the different effect of nucleotides, glutathione disulphide, sodium dodecyl sulfate and cations on the catalytic activity.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Sequence
  • Chromatography, DEAE-Cellulose
  • Chromatography, Gel
  • Cysteine Endopeptidases / isolation & purification
  • Endopeptidases / blood
  • Endopeptidases / isolation & purification*
  • Erythrocytes / enzymology*
  • Hemin / pharmacology
  • Humans
  • Isoelectric Point
  • Isoenzymes / antagonists & inhibitors
  • Isoenzymes / blood
  • Isoenzymes / isolation & purification*
  • Molecular Sequence Data
  • Multienzyme Complexes / isolation & purification
  • Oligopeptides / pharmacology
  • Peptides / metabolism
  • Proteasome Endopeptidase Complex
  • Substrate Specificity
  • Sulfhydryl Compounds / pharmacology

Substances

  • Isoenzymes
  • Multienzyme Complexes
  • Oligopeptides
  • Peptides
  • Sulfhydryl Compounds
  • Hemin
  • chymostatin
  • Endopeptidases
  • Cysteine Endopeptidases
  • Proteasome Endopeptidase Complex