Anti-inflammatory activity on LPS-stimulated dendritic cells of lupanetype triterpenoids from the leaves of Acanthopanax koreanum

Arch Pharm Res. 2011 Oct;34(10):1593-8. doi: 10.1007/s12272-011-1002-6. Epub 2011 Nov 12.

Abstract

Acanthopanax koreanum is well known herb in traditional Korean, Chinese, and Japanese anti-inflammatory action without any adverse effects. In the current study, we investigated the inhibitory effects of isolated compounds 1-13 from the leaves of A. koreanum on the lipopolysaccharide-stimulated production of pro-inflammatory cytokines in bone marrow-derived dendritic cells. Of these lupane-type triterpenoids, 1 exhibited particularly high inhibitory effect on lipopolysaccharide-stimulated TNF-α, IL-6, and IL-12 production with the values ranging from 45.0 to 84.5% at a concentration of 50 μM. These results warrant further studies concerning the potential anti-inflammatory benefits of medicinal foods containing the leaves of A. koreanum.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Anti-Inflammatory Agents, Non-Steroidal / pharmacology*
  • Bone Marrow Cells / drug effects
  • Cells, Cultured
  • Cytokines / biosynthesis
  • Dendritic Cells / drug effects*
  • Eleutherococcus / chemistry*
  • Interleukin-12 / biosynthesis
  • Interleukin-6 / biosynthesis
  • Lipopolysaccharides / pharmacology*
  • Mice
  • Mice, Inbred C57BL
  • Plant Extracts / chemistry
  • Plant Extracts / pharmacology
  • Plant Leaves / chemistry
  • Tetrazolium Salts
  • Thiazoles
  • Triterpenes / chemistry
  • Triterpenes / pharmacology*
  • Tumor Necrosis Factor-alpha / biosynthesis

Substances

  • Anti-Inflammatory Agents, Non-Steroidal
  • Cytokines
  • Interleukin-6
  • Lipopolysaccharides
  • Plant Extracts
  • Tetrazolium Salts
  • Thiazoles
  • Triterpenes
  • Tumor Necrosis Factor-alpha
  • Interleukin-12
  • lupane
  • thiazolyl blue