Anti-tumor-promoting activity of derivatives of abieslactone, a natural triterpenoid isolated from several Abies genus

Cancer Lett. 1990 Sep;53(2-3):141-4. doi: 10.1016/0304-3835(90)90206-d.

Abstract

Abiesenonic acid methyl ester (AVB-I acid methyl ester), a triterpenoid compound prepared from abieslactone, suppressed tumor promoter-induced phenomena in vitro and in vivo; i.e., AVB-I acid methyl ester inhibited 12-o-tetradecanoylphorbol-13-acetate (TPA)-stimulated 32Pi-incorporation into phospholipids of cultured cells and the promoting action of TPA on skin tumor formation in mice initiated with 7,12-dimethylbenz[a]anthracene.

MeSH terms

  • Animals
  • Carcinogens / pharmacology*
  • Female
  • HeLa Cells / metabolism
  • Lactones / pharmacology*
  • Mice
  • Mice, Inbred ICR
  • Phospholipids / metabolism
  • Skin Neoplasms / chemically induced
  • Tetradecanoylphorbol Acetate / pharmacology*
  • Trees
  • Triterpenes / pharmacology*

Substances

  • Carcinogens
  • Lactones
  • Phospholipids
  • Triterpenes
  • abieslactone
  • Tetradecanoylphorbol Acetate