Antihypertensive effect of a fixed-dose combination of losartan/hydrochlorothiazide in patients with uncontrolled hypertension: a multicenter study

Clin Exp Nephrol. 2012 Apr;16(2):269-78. doi: 10.1007/s10157-011-0564-4. Epub 2011 Nov 30.

Abstract

Background: Achieving adequate blood pressure (BP) control often requires more than one antihypertensive agent. The purpose of this study was to determine whether a fixed-dose formulation of losartan (LOS) plus hydrochlorothiazide (HCTZ) (LOS/HCTZ) is effective in achieving a greater BP lowering in patients with uncontrolled hypertension.

Methods: The study was a prospective, multicenter, observational trial exploring the antihypertensive effect of a single tablet of LOS 50 mg/HCTZ 12.5 mg. A total of 228 patients whose BP had previously been treated with more than one antihypertensive agents without having achieved BP goal below 130/80 mmHg enrolled in the study.

Results: A significant decrease in systolic and diastolic BP was observed in both clinic and home measurement after switching from the previous treatment to LOS/HCTZ. There was a significant decrease in both B-type natriuretic peptide (BNP) and urinary albumin creatinine (Cr) excretion ratio (ACR), especially in patients with elevated values. In contrast, there was a significant increase in serum Cr concentration in conjunction with a decrease in estimated glomerular filtration rate (eGFR). Overall serum uric acid (UA) concentration increased, whereas in patients with hyperuricemia there was a significant reduction in this value.

Conclusion: Switching to LOS/HCTZ provides a greater reduction in clinic and home BP in patients with uncontrolled hypertension. This combination therapy may lead to cardio-, reno protection and improve UA metabolism.

Publication types

  • Multicenter Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adult
  • Aged
  • Antihypertensive Agents / therapeutic use*
  • Blood Pressure / drug effects*
  • Blood Pressure Determination
  • Creatinine / urine
  • Drug Combinations
  • Female
  • Glomerular Filtration Rate
  • Humans
  • Hydrochlorothiazide / therapeutic use*
  • Hypertension / drug therapy*
  • Hypertension / metabolism
  • Hypertension / physiopathology
  • Hyperuricemia
  • Japan
  • Losartan / therapeutic use*
  • Male
  • Middle Aged
  • Natriuretic Peptide, Brain / blood
  • Prospective Studies
  • Treatment Outcome
  • Uric Acid / blood
  • Young Adult

Substances

  • Antihypertensive Agents
  • Drug Combinations
  • hydrochlorothiazide, losartan drug combination
  • Hydrochlorothiazide
  • Natriuretic Peptide, Brain
  • Uric Acid
  • Creatinine
  • Losartan