The role of the novel exopolyphosphatase MT0516 in Mycobacterium tuberculosis drug tolerance and persistence

PLoS One. 2011;6(11):e28076. doi: 10.1371/journal.pone.0028076. Epub 2011 Nov 21.

Abstract

Inorganic polyphosphate (poly P) has been postulated to play a regulatory role in the transition to bacterial persistence. In bacteria, poly P balance in the cell is maintained by the hydrolysis activity of the exopolyphosphatase PPX. However, the Mycobacterium tuberculosis PPX has not been characterized previously. Here we show that recombinant MT0516 hydrolyzes poly P, and an MT0516-deficient M. tuberculosis mutant exhibits elevated intracellular levels of poly P and increased expression of the genes mprB, sigE, and rel relative to the isogenic wild-type strain, indicating poly P-mediated signaling. Deficiency of MT0516 resulted in decelerated growth during logarithmic-phase in axenic cultures, and tolerance to the cell wall-active drug isoniazid. The MT0516-deficient mutant showed a significant survival defect in activated human macrophages and reduced persistence in the lungs of guinea pigs. We conclude that exopolyphosphatase is required for long-term survival of M. tuberculosis in necrotic lung lesions.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Acid Anhydride Hydrolases / deficiency
  • Acid Anhydride Hydrolases / metabolism*
  • Animals
  • Anti-Bacterial Agents / pharmacology
  • Bacterial Proteins / metabolism*
  • DNA Transposable Elements / genetics
  • Drug Resistance, Bacterial / drug effects*
  • Female
  • Genetic Complementation Test
  • Guinea Pigs
  • Humans
  • Hydrolysis / drug effects
  • Isoniazid / pharmacology*
  • Lung / drug effects
  • Lung / microbiology
  • Lung / pathology
  • Models, Molecular
  • Mutation / genetics
  • Mycobacterium tuberculosis / drug effects*
  • Mycobacterium tuberculosis / enzymology*
  • Mycobacterium tuberculosis / growth & development
  • Mycobacterium tuberculosis / pathogenicity
  • Polyphosphates / metabolism
  • Recombination, Genetic / genetics
  • Structural Homology, Protein
  • Virulence / drug effects

Substances

  • Anti-Bacterial Agents
  • Bacterial Proteins
  • DNA Transposable Elements
  • Polyphosphates
  • Acid Anhydride Hydrolases
  • exopolyphosphatase
  • Isoniazid