Resveratrol inhibits mucin gene expression, production and secretion from airway epithelial cells

Phytother Res. 2012 Jul;26(7):1082-7. doi: 10.1002/ptr.3701. Epub 2011 Dec 30.

Abstract

The study investigated whether resveratrol significantly affects mucin gene expression, production and secretion from airway epithelial cells. Confluent NCI-H292 cells were pretreated with resveratrol for 30 min and then stimulated with EGF (epidermal growth factor), PMA (phorbol 12-myristate 13-acetate) and TNF-α (tumor necrosis factor-α) for 24 h, respectively. The MUC5AC gene expression and mucin protein production were measured by RT-PCR and ELISA. The effect of resveratrol on TNF-α- or PMA-induced activation of NF-κB p65 was also examined. Confluent primary rat tracheal surface epithelial (RTSE) cells were pretreated with adenosine triphosphate (ATP) for 5 min and then treated for 30 min in the presence of resveratrol to assess the effect on mucin secretion using ELISA. The results were as follows: (1) resveratrol inhibited the expression of MUC5AC gene induced by EGF or PMA or TNF-α from NCI-H292 cells; (2) resveratrol also inhibited the production of MUC5AC mucin protein induced by the same inducers from NCI-H292 cells; (3) resveratrol inhibited the activation of NF-κB p65 by TNF-α or PMA in NCI-H292 cells; (4) resveratrol significantly decreased ATP-induced mucin secretion from cultured RTSE cells. This result suggests that resveratrol can regulate mucin gene expression, production and secretion, by directly acting on airway epithelial cells.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Cell Line
  • Epidermal Growth Factor / pharmacology
  • Epithelial Cells / drug effects*
  • Gene Expression / drug effects*
  • Humans
  • Male
  • Mucin 5AC / genetics
  • Mucin 5AC / metabolism*
  • Rats
  • Rats, Sprague-Dawley
  • Respiratory Mucosa / cytology
  • Resveratrol
  • Stilbenes / pharmacology*
  • Tetradecanoylphorbol Acetate / pharmacology
  • Trachea / cytology
  • Transcription Factor RelA / metabolism
  • Tumor Necrosis Factor-alpha / pharmacology

Substances

  • MUC5AC protein, human
  • Muc5ac protein, rat
  • Mucin 5AC
  • Stilbenes
  • Transcription Factor RelA
  • Tumor Necrosis Factor-alpha
  • Epidermal Growth Factor
  • Tetradecanoylphorbol Acetate
  • Resveratrol