Inhibition of neuroblastoma cell proliferation with omega-3 fatty acids and treatment of a murine model of human neuroblastoma using a diet enriched with omega-3 fatty acids in combination with sunitinib

Pediatr Res. 2012 Feb;71(2):168-78. doi: 10.1038/pr.2011.28. Epub 2011 Dec 21.

Abstract

Introduction: We investigated the use of dietary omega-3 (ω-3) polyunsaturated fatty acids (PUFAs) in the treatment of neuroblastoma both as a sole agent and in combination with sunitinib, a broad-spectrum tyrosine kinase receptor inhibitor.

Results: Substitution of all dietary fat with menhaden oil (ω-3 PUFA rich) resulted in a 40-70% inhibition of tumor growth and a statistically significant difference in the levels of several PUFAs (18:2 ω-6, 20:4 ω-6, 22:4 ω-6, 20:5 ω-3) as compared with a control diet. Furthermore, tumors from animals on the ω-3 fatty acid (FA)-enriched diet had an elevated triene/tetraene ratio suggestive of a change in local eicosanoid metabolism in these tissues similar to that seen with essential fatty acid deficiency. The ω-3 FA-enriched diet also decreased tumor-associated inflammatory cells and induced mitochondrial changes suggestive of mitochondrial damage. Combination treatment with sunitinib resulted in further reduction in tumor proliferation and microvessel density.

Discussion: These findings suggest a potential role for ω-3 PUFAs in the combination treatment of neuroblastoma.

Methods: We used a murine model of orthotopic and subcutaneous human neuroblastoma and diets that differ in the FA content to define the optimal dietary ω-3/omega-6 (ω-6) FA ratio required for the inhibition of these tumors.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Angiogenesis Inhibitors / pharmacology*
  • Animals
  • Arachidonic Acid / metabolism
  • Cell Line, Tumor
  • Cell Proliferation / drug effects*
  • Diet*
  • Dose-Response Relationship, Drug
  • Fatty Acids, Omega-3 / administration & dosage*
  • Fatty Acids, Omega-3 / metabolism
  • Fish Oils / administration & dosage*
  • Fish Oils / metabolism
  • Humans
  • Indoles / pharmacology*
  • Lipid Metabolism
  • Male
  • Mice
  • Mice, SCID
  • Microvessels / drug effects
  • Microvessels / pathology
  • Mitochondria / drug effects
  • Mitochondria / pathology
  • Neuroblastoma / blood supply
  • Neuroblastoma / diet therapy*
  • Neuroblastoma / drug therapy*
  • Neuroblastoma / enzymology
  • Neuroblastoma / pathology
  • Protein Kinase Inhibitors / pharmacology*
  • Pyrroles / pharmacology*
  • Sunitinib
  • Time Factors
  • Tumor Burden / drug effects
  • Xenograft Model Antitumor Assays

Substances

  • Angiogenesis Inhibitors
  • Fatty Acids, Omega-3
  • Fish Oils
  • Indoles
  • Protein Kinase Inhibitors
  • Pyrroles
  • Menhaden oil
  • Arachidonic Acid
  • Sunitinib