Effects of an agonist interleukin-2/Fc fusion protein, a mutant antagonist interleukin-15/Fc fusion protein, and sirolimus on cardiac allograft survival in non-human primates

J Heart Lung Transplant. 2012 Apr;31(4):427-35. doi: 10.1016/j.healun.2012.01.864. Epub 2012 Feb 24.

Abstract

Background: To tilt the immunologic balance toward tolerance and away from rejection, non-human primate recipients of cardiac allografts were treated with interleukin (IL)-2/Fc, mutant (m) antagonist type mIL-15/Fc, and sirolimus.

Methods: Heterotopic heart transplants were performed on 8 fully mismatched cynomolgus macaques. An untreated control recipient rejected its graft by post-operative Day 6. The remaining 7 animals received oral or intramuscular immunosuppression with sirolimus. A recipient treated with sirolimus alone rejected at the end of 28 days of immunosuppression. The remaining 6 monkeys also received IL-2/Fc and mIL-15/Fc intramuscularly until 28 days after transplant. One animal received a second 28-day course of fusion protein starting at Day 50. In these 6 animals, sirolimus was continued for 28 days (n = 4) or until protein levels were low (n = 2).

Results: In the 4 monkeys treated with a 28-day course of sirolimus and fusion proteins, mean graft survival was 51.5 days (range, 28-76 days). The animal receiving a second course of fusion protein rejected its graft on Day 177, despite detectable levels of the fusion proteins and sirolimus. The central memory, effector memory, and naïve CD4(+) and CD8(+) T-cell populations in the peripheral blood did not change significantly during fusion protein administration. A 2.5-fold expansion in CD4(+)CD25(+) lymphocytes occurred in recipients treated with fusion proteins and sirolimus that was not observed in the recipient treated with sirolimus alone.

Conclusions: Although IL-2/Fc, mIL-15/Fc, and sirolimus administered in this manner permitted modest prolongation of graft survival and expansion of CD4(+)CD25(+) T cells, tolerance was not achieved.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Biopsy
  • CD4-Positive T-Lymphocytes / immunology
  • CD4-Positive T-Lymphocytes / pathology
  • Graft Survival / drug effects*
  • Heart Transplantation / immunology*
  • Humans
  • Immunoglobulin Fc Fragments / pharmacology*
  • Immunosuppressive Agents / pharmacology
  • Interleukin-15 / pharmacology*
  • Interleukin-2 / pharmacology*
  • Interleukin-2 Receptor alpha Subunit / metabolism
  • Macaca fascicularis / immunology*
  • Models, Animal
  • Myocardium / immunology
  • Myocardium / pathology
  • Phenotype
  • Recombinant Fusion Proteins / pharmacology
  • Sirolimus / pharmacology*
  • Transplantation, Homologous

Substances

  • Immunoglobulin Fc Fragments
  • Immunosuppressive Agents
  • Interleukin-15
  • Interleukin-2
  • Interleukin-2 Receptor alpha Subunit
  • Recombinant Fusion Proteins
  • Sirolimus