3,4-methylenedioxymethamphetamine (ecstasy) decreases inflammation and airway reactivity in a murine model of asthma

Neuroimmunomodulation. 2012;19(4):209-19. doi: 10.1159/000334098. Epub 2012 Mar 21.

Abstract

Objective: 3,4-Methylenedioxymethamphetamine (MDMA), or ecstasy, is a synthetic drug used recreationally, mainly by young people. It has been suggested that MDMA has a Th cell skewing effect, in which Th1 cell activity is suppressed and Th2 cell activity is increased. Experimental allergic airway inflammation in ovalbumin (OVA)-sensitized rodents is a useful model to study Th2 response; therefore, based on the Th2 skewing effect of MDMA, we studied MDMA in a model of allergic lung inflammation in OVA-sensitized mice.

Methods: We evaluated cell trafficking in the bronchoalveolar lavage fluid, blood and bone marrow; cytokine production; L-selectin expression and lung histology. We also investigated the effects of MDMA on tracheal reactivity in vitro and mast cell degranulation.

Results: We found that MDMA given prior to OVA challenge in OVA-sensitized mice decreased leukocyte migration into the lung, as revealed by a lower cell count in the bronchoalveolar lavage fluid and lung histologic analysis. We also showed that MDMA decreased expression of both Th2-like cytokines (IL-4, IL-5 and IL-10) and adhesion molecules (L-selectin). Moreover, we showed that the hypothalamus-pituitary-adrenal axis is partially involved in the MDMA-induced reduction in leukocyte migration into the lung. Finally, we showed that MDMA decreased tracheal reactivity to methacholine as well as mast cell degranulation in situ.

Conclusions: Thus, we report here that MDMA given prior to OVA challenge in OVA-sensitized allergic mice is able to decrease lung inflammation and airway reactivity and that hypothalamus-pituitary-adrenal axis activation is partially involved. Together, the data strongly suggest an involvement of a neuroimmune mechanism in the effects of MDMA on lung inflammatory response and cell recruitment to the lungs of allergic animals.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Asthma / immunology*
  • Bone Marrow Cells
  • Bronchoalveolar Lavage Fluid / cytology
  • Cell Movement / drug effects
  • Cytokines / drug effects
  • Cytokines / metabolism
  • Disease Models, Animal
  • Inflammation / immunology*
  • Leukocyte Count
  • Leukocytes / drug effects*
  • Lung / cytology
  • Lung / drug effects*
  • Male
  • Mast Cells / drug effects
  • Mice
  • N-Methyl-3,4-methylenedioxyamphetamine / immunology
  • N-Methyl-3,4-methylenedioxyamphetamine / pharmacology*
  • Th2 Cells / drug effects*
  • Th2 Cells / physiology
  • Trachea / drug effects

Substances

  • Cytokines
  • N-Methyl-3,4-methylenedioxyamphetamine