Regulation of SIRT1 activity by genotoxic stress

Genes Dev. 2012 Apr 15;26(8):791-6. doi: 10.1101/gad.188482.112. Epub 2012 Mar 30.

Abstract

SIRT1 regulates a variety of cellular functions, including cellular stress responses and energy metabolism. SIRT1 activity is negatively regulated by DBC1 (Deleted in Breast Cancer 1) through direct binding. However, how the DBC1-SIRT1 interaction is regulated remains unclear. We found that the DBC1-SIRT1 interaction increases following DNA damage and oxidative stress. The stress-induced DBC1-SIRT1 interaction requires the ATM-dependent phosphorylation of DBC1 at Thr 454, which creates a second binding site for SIRT1. Finally, we showed that the stress-induced DBC1-SIRT1 interaction is important for cell fate determination following genotoxic stress. These results revealed a novel mechanism of SIRT1 regulation during genotoxic stress.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Adaptor Proteins, Signal Transducing
  • Ataxia Telangiectasia Mutated Proteins
  • Binding Sites
  • Cell Cycle Proteins / metabolism
  • Cell Line, Tumor
  • DNA-Binding Proteins / metabolism
  • Humans
  • Phosphorylation
  • Protein Serine-Threonine Kinases / metabolism
  • Sirtuin 1 / genetics
  • Sirtuin 1 / metabolism*

Substances

  • Adaptor Proteins, Signal Transducing
  • CCAR2 protein, human
  • Cell Cycle Proteins
  • DNA-Binding Proteins
  • ATM protein, human
  • Ataxia Telangiectasia Mutated Proteins
  • Protein Serine-Threonine Kinases
  • SIRT1 protein, human
  • Sirtuin 1