Effects of gut-targeted 15-LOX-1 transgene expression on colonic tumorigenesis in mice

J Natl Cancer Inst. 2012 May 2;104(9):709-16. doi: 10.1093/jnci/djs187. Epub 2012 Apr 2.

Abstract

Expression of 15-lipoxygenase-1 (15-LOX-1) is decreased in many human cancers; however, the mechanistic significance of its decreased expression has been difficult to determine because its mouse homolog 12/15-LOX has opposing functions. We generated a mouse model in which expression of a human 15-LOX-1 transgene was targeted to the intestinal epithelium via the villin promoter. Targeted expression was confirmed by real-time reverse transcription-polymerase chain reaction and immunoblotting. When the 15-LOX-1 transgene was expressed in colonic epithelial cells of two independent mouse lines (B6 and FVB), azoxymethane-inducible colonic tumorigenesis was suppressed (mean number of tumors: wild type [WT] = 8.2, 15-LOX-1(+/-) = 4.91, 15-LOX-1(+/+) = 3.57; WT vs 15-LOX-1(+/-) two-sided P = .003, WT vs 15-LOX-1(+/+) two-sided P < .001; n = 10-14 mice per group). 15-LOX-1 transgene expression was always decreased in the tumors that did develop. In the presence of expression of the 15-LOX-1 transgene, expression of tumor necrosis factor alpha and its target inducible nitric oxide synthase were decreased and activation of nuclear factor-kappa B in colonic epithelial cells was inhibited.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Arachidonate 15-Lipoxygenase / genetics*
  • Arachidonate 15-Lipoxygenase / metabolism*
  • Azoxymethane
  • Carcinogens
  • Cell Transformation, Neoplastic / genetics
  • Cell Transformation, Neoplastic / metabolism
  • Colon / enzymology*
  • Colonic Neoplasms / chemically induced
  • Colonic Neoplasms / enzymology*
  • Disease Models, Animal
  • Epithelial Cells / enzymology
  • Gene Expression Regulation, Enzymologic
  • Gene Expression Regulation, Neoplastic
  • Immunoblotting
  • Intestinal Mucosa / enzymology*
  • Mice
  • Mice, Transgenic
  • NF-kappa B / metabolism
  • Nitric Oxide Synthase Type II / metabolism
  • RNA, Messenger / metabolism
  • Real-Time Polymerase Chain Reaction
  • Transgenes*
  • Tumor Necrosis Factor-alpha / metabolism
  • Up-Regulation

Substances

  • Carcinogens
  • NF-kappa B
  • RNA, Messenger
  • Tumor Necrosis Factor-alpha
  • Arachidonate 15-Lipoxygenase
  • Nitric Oxide Synthase Type II
  • Azoxymethane