Molecular mechanisms that desensitize metabotropic glutamate receptor signaling: an overview

Neuropharmacology. 2013 Mar:66:24-30. doi: 10.1016/j.neuropharm.2012.05.005. Epub 2012 May 29.

Abstract

The purpose of the present article is to review our actual knowledge on the desensitization of metabotropic glutamate receptors based on the literature available so far, with the attempt to emphasize all converging data and to give a possible explanation to those evidences that still remain controversial. 1. We review our knowledge on the regulation of mGlu receptors based on the available literature 2. We report converging data and we comment on issues that still remain controversial. This article is part of a Special Issue entitled 'Metabotropic Glutamate Receptors'.

Publication types

  • Review

MeSH terms

  • Animals
  • Cyclic AMP / antagonists & inhibitors
  • Cyclic AMP / biosynthesis
  • Extracellular Signal-Regulated MAP Kinases / drug effects
  • Extracellular Signal-Regulated MAP Kinases / metabolism
  • Humans
  • Receptors, Metabotropic Glutamate / metabolism*
  • Signal Transduction / drug effects*

Substances

  • Receptors, Metabotropic Glutamate
  • Cyclic AMP
  • Extracellular Signal-Regulated MAP Kinases