Comparison of sister-chromatid exchange frequencies in mouse T- and B-lymphocytes after exposure to 4-hydroxycyclophosphamide or phosphoramide mustard

Mutat Res. 1990 Dec;245(4):293-7. doi: 10.1016/0165-7992(90)90159-h.

Abstract

The present study was designed to investigate the genotoxicity of 4-hydroxycyclophosphamide (4-OHCP) and phosphoramide mustard (PAM), both reactive metabolites of cyclophosphamide (CP), for possible differences in SCE-inducing activity in mouse T- and B-lymphocytes. Mouse peripheral blood lymphocytes were isolated and stimulated to divide with either phytohemagglutinin (T-cell mitogen) or lipopolysaccharide (a polyclonal B-cell activator). Significant concentration-dependent increases in SCE frequencies were observed for both 4-OHCP and PAM with both mitogens, with 4-OHCP being almost twice as potent as PAM. There was no difference in SCE response between T- and B-lymphocytes after exposure to either PAM or 4-OHCP. These data do not support the idea that the difference in SCE response in T- and B-lymphocytes by CP in vivo is due to differential responses to either of the proposed putative metabolites of CP.

MeSH terms

  • Animals
  • B-Lymphocytes / drug effects*
  • B-Lymphocytes / metabolism*
  • B-Lymphocytes / ultrastructure
  • Cells, Cultured
  • Cyclophosphamide / analogs & derivatives*
  • Cyclophosphamide / toxicity
  • Lipopolysaccharides / pharmacology
  • Male
  • Mice
  • Mice, Inbred C57BL
  • Mutagenicity Tests
  • Phosphoramide Mustards / toxicity*
  • Phytohemagglutinins / pharmacology
  • Sister Chromatid Exchange*
  • T-Lymphocytes / drug effects*
  • T-Lymphocytes / metabolism
  • T-Lymphocytes / ultrastructure

Substances

  • Lipopolysaccharides
  • Phosphoramide Mustards
  • Phytohemagglutinins
  • phosphoramide mustard
  • 4-hydroxycyclophosphamide
  • Cyclophosphamide