Structural and thermodynamic characterization of the self-adhesive properties of human P-cadherin

Mol Biosyst. 2012 Aug;8(8):2050-3. doi: 10.1039/c2mb25161b. Epub 2012 Jun 7.

Abstract

Human P-cadherin is a promising therapeutic target against cancer. However, its characterization at the molecular level is still lacking. We report that human P-cadherin associated irreversibly in a distinct dimer configuration. Unexpectedly, the divalent cation Ca²⁺ was not necessary for dimerization, although it greatly stabilized the protein-protein complex.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Cadherins / chemistry*
  • Cadherins / metabolism*
  • Calcium / chemistry*
  • Calcium / metabolism*
  • Dimerization
  • Humans
  • Models, Biological
  • Protein Binding
  • Protein Structure, Tertiary
  • Thermodynamics

Substances

  • Cadherins
  • Calcium