Decreasing herpes simplex viral infectivity in solution by surface-immobilized and suspended N,N-dodecyl,methyl-polyethylenimine

Pharm Res. 2013 Jan;30(1):25-31. doi: 10.1007/s11095-012-0825-2. Epub 2012 Jul 14.

Abstract

Purpose: To explore surface-immobilized and suspended modalities of the hydrophobic polycation N,N-dodecyl,methyl-polyethylenimine (DMPEI) for the ability to reduce viral infectivity in aqueous solutions containing herpes simplex viruses (HSVs) 1 and 2.

Methods: Surface-immobilized (coated onto surfaces) and suspended DMPEI were incubated with aqueous solutions containing HSV-1 or -2 to measure the antiviral effect of the hydrophobic polycation's formulations on HSVs.

Results: DMPEI coated on either polyethylene slides or male latex condoms dramatically decreases infectivity in solutions containing HSV-1 or -2. Moreover, DMPEI suspended in aqueous solution markedly reduces the infectious titer of these HSVs.

Conclusion: Our results suggest potential uses of DMPEI for both prophylaxis (in the form of coated condoms) and treatment (as a topical suspension) for HSV infections.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Antiviral Agents / administration & dosage
  • Antiviral Agents / therapeutic use*
  • Condoms / virology
  • Herpes Genitalis / prevention & control
  • Herpes Genitalis / transmission*
  • Herpes Genitalis / virology
  • Herpes Simplex / prevention & control
  • Herpes Simplex / transmission*
  • Herpes Simplex / virology
  • Herpesvirus 1, Human / drug effects
  • Herpesvirus 1, Human / pathogenicity*
  • Herpesvirus 2, Human / drug effects
  • Herpesvirus 2, Human / pathogenicity*
  • Humans
  • Male
  • Polyethyleneimine / administration & dosage
  • Polyethyleneimine / analogs & derivatives*
  • Polyethyleneimine / therapeutic use
  • Surface Properties

Substances

  • Antiviral Agents
  • N,N-dodecyl,methyl-polyethylenimine
  • Polyethyleneimine