An antithrombin-heparin complex increases the anticoagulant activity of fibrin clots

Res Lett Biochem. 2008:2008:639829. doi: 10.1155/2008/639829. Epub 2008 Apr 14.

Abstract

Clotting blood contains fibrin-bound thrombin, which is a major source of procoagulant activity leading to clot extension and further activation of coagulation. When bound to fibrin, thrombin is protected from inhibition by antithrombin (AT) + heparin but is neutralized when AT and heparin are covalently linked (ATH). Here, we report the surprising observation that, rather than yielding an inert complex, thrombin-ATH formation converts clots into anticoagulant surfaces that effectively catalyze inhibition of thrombin in the surrounding environment.