Age effects on serotonin receptor 1B as assessed by PET

J Nucl Med. 2012 Sep;53(9):1411-4. doi: 10.2967/jnumed.112.103598. Epub 2012 Jul 31.

Abstract

Previous imaging studies have suggested that there is an age-related decline in brain serotonin (5-hydroxytryptamine) measures in healthy subjects. This paper addresses whether the availability of 5-hydroxytryptamine receptor 1B (5-HT(1B)) is seen to decrease with aging via PET imaging.

Methods: Forty-eight healthy control subjects (mean age ± SD, 30 ± 10 y; age range, 18-61 y; 33 men, 15 women) underwent (11)C-P943 scanning on a high-resolution PET tomograph. Regions were examined with and without gray matter masking, the latter in an attempt to control for age-related gray matter atrophy on nondisplaceable binding potential (BP(ND)) as determined by a validated multilinear reference tissue model.

Results: 5-HT(1B) BP(ND) decreased in the cortex at an average rate of 8% per decade without and 9% with gray matter masking. A negative association with age was also observed in all individual cortical regions. Differences in the putamen and pallidum (positive association) were significant after adjustment for multiple comparisons. No sex- or race-related effects on 5-HT(1B) BP(ND) were found in any regions.

Conclusion: These findings indicate that age is a relevant factor for 5-HT(1B) in the cortex of healthy adults.

Publication types

  • Clinical Trial
  • Research Support, American Recovery and Reinvestment Act
  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adolescent
  • Adult
  • Aging / metabolism*
  • Carbon Radioisotopes
  • Cerebral Cortex / diagnostic imaging
  • Cerebral Cortex / metabolism
  • Female
  • Humans
  • Ligands
  • Male
  • Middle Aged
  • Piperazines / metabolism
  • Positron-Emission Tomography*
  • Pyrrolidinones / metabolism
  • Receptor, Serotonin, 5-HT1B / metabolism*
  • Substrate Specificity
  • Young Adult

Substances

  • 1-(4-(2-methoxyisopropyl)phenyl)-3-(2-(4-methylpiperazin-1-yl)benzyl)pyrrolidin-2-one
  • Carbon Radioisotopes
  • Ligands
  • Piperazines
  • Pyrrolidinones
  • Receptor, Serotonin, 5-HT1B