Identification of hepatocyte growth factor activator (Hgfac) gene as a target of HNF1α in mouse β-cells

Biochem Biophys Res Commun. 2012 Aug 31;425(3):619-24. doi: 10.1016/j.bbrc.2012.07.134. Epub 2012 Aug 1.

Abstract

HNF1α is a transcription factor that is expressed in pancreatic β-cells and mutations of the HNF1α gene cause a form of monogenic diabetes. To understand the role of HNF1α in pancreatic β-cells, we established the MIN6 β-cell line that stably expressed HNF1α-specific shRNA. Expression of the gene encoding hepatocyte growth factor (HGF) activator (Hgfac), a serine protease that efficiently activates HGF, was decreased in HNF1α KD-MIN6 cells. Down-regulation of Hgfac expression was also found in the islets of HNF1α (+/-) mice. Reporter gene analysis and the chromatin immunoprecipitation assay indicated that HNF1α directly regulates the expression of Hgfac in β-cells. It has been reported that HGF has an important influence on β-cell mass and β-cell function. Thus, HNF1α might regulate β-cell mass or function at least partly by modulating Hgfac expression.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Base Sequence
  • Cell Line
  • Gene Expression Regulation*
  • Hepatocyte Nuclear Factor 1-alpha / genetics
  • Hepatocyte Nuclear Factor 1-alpha / metabolism*
  • Humans
  • Insulin-Secreting Cells / metabolism*
  • Mice
  • Molecular Sequence Data
  • Oligonucleotide Array Sequence Analysis
  • RNA, Small Interfering / genetics
  • Serine Endopeptidases / genetics*

Substances

  • Hepatocyte Nuclear Factor 1-alpha
  • Hnf1a protein, mouse
  • RNA, Small Interfering
  • HGF activator
  • Serine Endopeptidases