The growth of the canine glioblastoma cell line D-GBM and the canine histiocytic sarcoma cell line DH82 is inhibited by the resveratrol oligomers hopeaphenol and r2-viniferin

Vet Comp Oncol. 2014 Jun;12(2):149-59. doi: 10.1111/j.1476-5829.2012.00349.x. Epub 2012 Aug 10.

Abstract

Vineatrol(®) 30 is a grapevine-shoot extract, which contains resveratrol as well as considerable amounts of so-called resveratrol oligomers such as hopeaphenol and r2-viniferin. In this study, we analysed whether the two above-mentioned resveratrol oligomers were able to inhibit the growth of the canine glioblastoma cell line D-GBM and the canine histiocytic sarcoma cell line DH82, compared their potency to inhibit tumour cell growth with that of resveratrol and determined whether the induction of apoptosis via caspase 9 and 3/7 activation underlies the tumour cell growth-inhibiting effect of hopeaphenol and r2-viniferin. Vineatrol(®) 30, resveratrol, hopeaphenol and r2-viniferin inhibited the growth of D-GBM and DH82 cells in a concentration-dependent manner, whereby hopeaphenol and r2-viniferin were more potent than resveratrol itself in inhibiting the growth of the canine tumour cell lines. Moreover, the anti-proliferative effect of both resveratrol oligomers in D-GBM cells is based on their capacity to induce caspase 9 and 3/7 activation.

Keywords: apoptosis; canine tumour cell lines; glioblastoma; histiocytic sarcoma; resveratrol; resveratrol oligomers.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Antineoplastic Agents / chemistry
  • Antineoplastic Agents / pharmacology
  • Cell Line, Tumor
  • Dogs*
  • Glioblastoma / metabolism*
  • Histiocytic Sarcoma / metabolism*
  • Molecular Structure
  • Phenols
  • Polyphenols / chemistry*
  • Polyphenols / pharmacology
  • Resveratrol
  • Stilbenes / chemistry*
  • Stilbenes / pharmacology*

Substances

  • Antineoplastic Agents
  • Phenols
  • Polyphenols
  • Stilbenes
  • hopeaphenol
  • r2-viniferin
  • Resveratrol