Fibroblast growth factor 23: state of the field and future directions

Trends Endocrinol Metab. 2012 Dec;23(12):610-8. doi: 10.1016/j.tem.2012.07.002. Epub 2012 Aug 24.

Abstract

Fibroblast growth factor 23 (FGF23) is a bone-derived hormone that regulates and is regulated by blood levels of phosphate and active vitamin D. Post-translational glycosylation by the enzyme GALNT3 and subsequent processing by furin have been demonstrated to be a regulated process that plays a role in regulating FGF23 levels. In physiologic states, FGF23 signaling is mediated by an FGF receptor and the coreceptor, Klotho. Recent work identifying a role for iron/hypoxia pathways in FGF23 physiology and their implications are discussed. Beyond its importance in primary disorders of mineral metabolism, recent work implicates FGF23 in renal disease-associated morbidity, as well as possible roles in cardiovascular disease and skeletal fragility.

Publication types

  • Research Support, N.I.H., Intramural
  • Review

MeSH terms

  • Animals
  • Bone and Bones / metabolism
  • Fibroblast Growth Factor-23
  • Fibroblast Growth Factors / physiology*
  • Glucuronidase / physiology
  • Humans
  • Iron Metabolism Disorders / physiopathology
  • Kidney Diseases / metabolism
  • Klotho Proteins
  • Mice
  • Receptors, Fibroblast Growth Factor / physiology
  • Vitamin D / physiology

Substances

  • FGF23 protein, human
  • Fgf23 protein, mouse
  • Receptors, Fibroblast Growth Factor
  • Vitamin D
  • Fibroblast Growth Factors
  • Fibroblast Growth Factor-23
  • Glucuronidase
  • Klotho Proteins