No effect of thioridazine on plasma concentrations of carbamazepine and its active metabolite carbamazepine-10,11-epoxide

Ther Drug Monit. 1990 Sep;12(5):511-3. doi: 10.1097/00007691-199009000-00017.

Abstract

The effect of an oral treatment with thioridazine (100 or 200 mg daily) on plasma concentrations of carbamazepine (CBZ) and its active metabolite carbamazepine-10,11-epoxide (CBZ-E) was studied in eight epileptic patients stabilized on CBZ therapy. No significant changes in steady-state plasma levels of CBZ and CBZ-E occurred, suggesting that CBZ metabolism is not apparently affected by thioridazine.

MeSH terms

  • Adult
  • Carbamazepine / analogs & derivatives*
  • Carbamazepine / blood*
  • Carbamazepine / therapeutic use
  • Epilepsy / blood
  • Epilepsy / drug therapy
  • Female
  • Homeostasis
  • Humans
  • Male
  • Middle Aged
  • Thioridazine / administration & dosage
  • Thioridazine / blood
  • Thioridazine / pharmacology*

Substances

  • Carbamazepine
  • Thioridazine
  • carbamazepine epoxide