Effect of LY294002 on adriamycin-induced epithelial-mesenchymal transition in human breast carcinoma cells

Zhongguo Yi Xue Ke Xue Yuan Xue Bao. 2012 Aug;34(4):319-23. doi: 10.3881/j.issn.1000-503X.2012.04.002.

Abstract

Objective: To study the effect of LY294002 on the adriamycin- induced epithelial-mesenchymal transition in human breast carcinoma cells.

Methods: Human breast carcinoma cells MCF-7 was cultured in vitro and then exposed to adriamycin with or without LY294002. The protein expression levels of Akt, phosphorylated-Akt (p-Akt), Snail, and E-cadherin was detected by Western blot analysis. The mRNA expressions of Snail and E-cadherin were determined by RT-PCR.

Results: Adriamycin significantly increased the protein expression of Snail and depressed the protein expression of E-cadherin (P<0.05). The pre-treatment with LY294002 significantly reversed the changes of activities and levels of the above proteins (P<0.05).

Conclusion: LY294002 could reverse the adriamycin-induced epithelial-mesenchymal transition in human breast carcinoma cells by regulating the expressions of Snail and E-cadherin through suppressing PI3K/Akt signaling pathway.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Antigens, CD
  • Breast Neoplasms / metabolism
  • Breast Neoplasms / pathology*
  • Cadherins / metabolism
  • Chromones / pharmacology*
  • Doxorubicin / pharmacology*
  • Epithelial-Mesenchymal Transition / drug effects*
  • Humans
  • MCF-7 Cells
  • Morpholines / pharmacology*
  • Phosphoinositide-3 Kinase Inhibitors
  • Proto-Oncogene Proteins c-akt / metabolism
  • Signal Transduction / drug effects*
  • Snail Family Transcription Factors
  • Transcription Factors / metabolism

Substances

  • Antigens, CD
  • CDH1 protein, human
  • Cadherins
  • Chromones
  • Morpholines
  • Phosphoinositide-3 Kinase Inhibitors
  • Snail Family Transcription Factors
  • Transcription Factors
  • 2-(4-morpholinyl)-8-phenyl-4H-1-benzopyran-4-one
  • Doxorubicin
  • Proto-Oncogene Proteins c-akt