New steroidal saponins from the bulbs of Lilium brownii var. viridulum

Carbohydr Res. 2012 Nov 1:361:19-26. doi: 10.1016/j.carres.2012.07.027. Epub 2012 Aug 8.

Abstract

Phytochemical investigation of the bulbs of Lilium brownii var. viridulum led to the isolation of seven new steroidal saponins (1-7), along with eight known analogues (8-15). The new steroidal saponins were identified as 27-O-[(3S)-3-O-β-D-glucopyranosyl 3-methylglutaroyl]isonarthogenin 3-O-[α-L-rhamnopyranosyl-(1→2)]-β-D-glucopyranoside (1), (24S,25S)-3β,17α,24-trihydroxy-5α-spirostan-6-one 3-O-[α-L-rhamnopyranosyl-(1→2)]-β-D-glucopyranoside (2), tenuifoliol 3-O-[β-D-glucopyranosyl-(1→4)]-β-D-glucopyranoside (3), 26-O-β-D-glucopyranosylnuatigenin (4), 26-O-β-D-glucopyranosylnuatigenin 3-O-β-D-glucopyranoside (5), 26-O-β-D-glucopyranosylnuatigenin 3-O-{α-L-rhamnopyranosyl-(1→2)-[β-D-glucopyranosyl-(1→6)]}-β-D-glucopyranoside (6), 26-O-[β-D-glucopyranosyl-(1→2)]-β-D-glucopyranosylnuatigenin 3-O-[α-L-rhamnopyranosyl-(1→2)]-β-D-glucopyranoside (7), using a combination of spectroscopic evidence and chemical methods. The carbohydrate chain of a sugar linked to C-3 of the HMG group (3-hydroxy-3-methylglutarate) in compound 1 is rarely found in nature. Compound 2 possesses a new (24S,25S)-3β,17α,24-trihydroxy-5α-spirostan-6-one aglycon moiety. The disaccharide chain linked to C-26 hydroxy group of the furospirostanol in compound 7 has not been observed from natural sources.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Cell Line
  • Dose-Response Relationship, Drug
  • Drug Evaluation, Preclinical
  • HeLa Cells
  • Hep G2 Cells
  • Humans
  • Hydrolysis
  • Lilium / chemistry*
  • Lipopolysaccharides / antagonists & inhibitors
  • Lipopolysaccharides / pharmacology
  • Macrophages / drug effects
  • Macrophages / metabolism
  • Mice
  • Molecular Conformation
  • Nitric Oxide / antagonists & inhibitors
  • Nitric Oxide / biosynthesis
  • Plant Roots / chemistry*
  • Saponins / isolation & purification*
  • Saponins / pharmacology
  • Stereoisomerism
  • Steroids / isolation & purification*
  • Steroids / pharmacology
  • Structure-Activity Relationship

Substances

  • Lipopolysaccharides
  • Saponins
  • Steroids
  • Nitric Oxide