The tail nick augments Aeromonas sobria serine protease (ASP) activity in plasma through retarding inhibition by α2-macroglobulin

FEBS Lett. 2012 Oct 19;586(20):3613-7. doi: 10.1016/j.febslet.2012.08.004. Epub 2012 Aug 14.

Abstract

ASP is a serine protease secreted by Aeromonas sobria, a sepsis-causing bacterium, and induces sepsis-mimicking disorders through plasma protein cleavage. The pathogen also secretes nASP that has a nick in the carboxy-terminal region. Compared with single-chain ASP (sASP), nASP had near-equivalent activity for small peptide substrates but was less proteolytic. Surprisingly, nASP cleaved proteins more in plasma and was inhibited by human α(2)-macroglobulin more slowly than sASP. Retarded inhibition by α(2)-macroglobulin allows nASP to keep proteolytic activity for longer in the host and exacerbate disorders at Aeromonas sobria infection sites. nASP may be an evolutional form to augment ASP virulence.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Aeromonas / enzymology*
  • Amino Acid Sequence
  • Catalytic Domain
  • Humans
  • Models, Molecular
  • Oligopeptides / chemistry
  • Oligopeptides / metabolism
  • Proteolysis / drug effects
  • Serine Proteases / blood
  • Serine Proteases / chemistry*
  • Serine Proteases / metabolism*
  • Serine Proteinase Inhibitors / pharmacology*
  • alpha-Macroglobulins / pharmacology*

Substances

  • Oligopeptides
  • Serine Proteinase Inhibitors
  • alpha-Macroglobulins
  • Serine Proteases