Unexpected mucin-type O-glycosylation and host-specific N-glycosylation of human recombinant interleukin-17A expressed in a human kidney cell line

Protein Expr Purif. 2013 Jan;87(1):27-34. doi: 10.1016/j.pep.2012.09.013. Epub 2012 Oct 13.

Abstract

The T helper cell-derived cytokine interleukin-17A (IL-17A) is a variably glycosylated disulfide-linked homodimer of 34-38 kDa. Its polypeptide monomer contains one canonical N-glycosylation site at Asn68, and human recombinant IL-17A was partly N-glycosylated when expressed in human kidney (HEK293) cells as a fusion protein with a melittin signal sequence and an N-terminal hexahistidine tag. Orbitrap mass analyses of the tryptic N-glycopeptide 63-69 indicated that the N-glycosylation was of the GalNAc-terminated type characteristic of cultured kidney cells. The mass spectrum of IL-17A monomer also included peaks shifted by +948 Da from the respective masses of unglycosylated and N-glycosylated polypeptides. These were caused by unpredicted partial O-glycosylation of Thr26 with the mucin-like structure -GalNAc(-NeuNAc)-Gal-NeuNAc. Identical O-glycosylation occurred in commercially sourced recombinant IL-17A also expressed in HEK293 cells but with a different N-terminal sequence. Therefore, the kidney host cell line not only imposed its characteristic pattern of N-glycosylation on recombinant IL-17A but additionally created an O-glycosylation not known to be present in the T cell-derived cytokine. Mammalian host cell lines for recombinant protein expression generally impose their characteristic patterns of N-glycosylation on the product, but this work exemplifies how a host may also unpredictably O-glycosylate a protein that is probably not normally O-glycosylated.

MeSH terms

  • Amino Acid Sequence
  • CD4-Positive T-Lymphocytes / metabolism
  • Carbohydrate Conformation
  • Carbohydrate Sequence
  • Glycosylation
  • HEK293 Cells
  • Humans
  • Insect Proteins / biosynthesis
  • Insect Proteins / chemistry
  • Interleukin-17 / biosynthesis*
  • Interleukin-17 / chemistry
  • Melitten / biosynthesis
  • Melitten / chemistry
  • Molecular Sequence Data
  • Molecular Weight
  • Peptide Mapping
  • Protein Processing, Post-Translational*
  • Protein Sorting Signals
  • Recombinant Fusion Proteins / biosynthesis*
  • Recombinant Fusion Proteins / chemistry
  • Tandem Mass Spectrometry

Substances

  • IL17A protein, human
  • Insect Proteins
  • Interleukin-17
  • Protein Sorting Signals
  • Recombinant Fusion Proteins
  • Melitten