Treatment of hepatitis C in patients infected with human immunodeficiency virus in the direct-acting antiviral era

Infect Dis Clin North Am. 2012 Dec;26(4):931-48. doi: 10.1016/j.idc.2012.08.004. Epub 2012 Sep 10.

Abstract

Chronic hepatitis C is a leading cause of clinical complications and mortality in individuals infected with human immunodeficiency virus (HIV). Approval for the first direct-acting antiviral (DAA) against the hepatitis C virus (HCV) has been eagerly awaited for treating patients coinfected with HIV/HCV. The use of first-generation HCV protease inhibitors is challenged by complicated dosing schedules, frequent serious toxicities, unwanted drug interactions, drug resistance, and high cost. First-generation DAAs will eventually be replaced by more potent, well-tolerated, and convenient agents. HIV/HCV co-infection will become restricted to individuals without proper access to health care.

MeSH terms

  • Antiviral Agents / therapeutic use*
  • Coinfection / drug therapy
  • Coinfection / virology
  • Drug Resistance, Viral
  • HIV Infections / drug therapy
  • HIV Infections / virology*
  • Hepacivirus / isolation & purification
  • Hepatitis C / drug therapy*
  • Hepatitis C / virology*
  • Humans
  • Oligopeptides / therapeutic use
  • Proline / analogs & derivatives
  • Proline / therapeutic use

Substances

  • Antiviral Agents
  • Oligopeptides
  • telaprevir
  • N-(3-amino-1-(cyclobutylmethyl)-2,3-dioxopropyl)-3-(2-((((1,1-dimethylethyl)amino)carbonyl)amino)-3,3-dimethyl-1-oxobutyl)-6,6-dimethyl-3-azabicyclo(3.1.0)hexan-2-carboxamide
  • Proline