Differential effects of heart rate reduction by atenolol or ivabradine on peripheral endothelial function in type 2 diabetic patients

Heart. 2012 Dec;98(24):1812-6. doi: 10.1136/heartjnl-2012-302795. Epub 2012 Oct 19.

Abstract

Objective: To assess whether reduction of heart rate (HR) has beneficial effects on endothelial function in patients with type 2 diabetes mellitus (T2DM).

Design: Randomised, double-blind, placebo-controlled study.

Setting: University hospital.

Patients: 66 T2DM patients without overt cardiovascular disease.

Interventions: Patients were randomised to receive for 4 weeks, in addition to their standard therapy, one of the following treatments: atenolol (25 mg twice daily), ivabradine (5 mg twice daily) or placebo (1 tablet twice daily).

Main outcome measures: Systemic endothelial function, assessed by flow-mediated dilation (FMD); endothelium-independent vasodilation, assessed by nitrate-mediated dilation (NMD); cardiac autonomic function, assessed by HR variability (HRV).

Results: 61 patients completed the study (19, 22 and 20 patients in atenolol, ivabradine and placebo groups, respectively). Compared with baseline, HR was similarly reduced by atenolol (87±13 vs 69±9 bpm) and ivabradine (86±12 to 71±9 bpm), but not by placebo (82±10 vs 81±9 bpm) (p<0.001). FMD improved at follow-up in the atenolol group (4.8±1.7 vs 6.4±1.9%), but not in the ivabradine group (5.2±2.5 vs 4.9±2.2%) and in the placebo group (4.8±1.5 vs 4.7±1.7%) (p<0.01). NMD did not change significantly in any group. HRV parameters did not change in the placebo group; they, instead, consistently increased in the atenolol, whereas a mild increase in SDNNi was only observed in the ivabradine group. A significant correlation was found in the atenolol group between HR and FMD changes (r=-0.48; p=0.04).

Conclusions: Despite a comparable reduction in HR, atenolol, but not ivabradine, improved FMD in T2DM patients suggesting that changes in HR are by themselves unlikely to significantly improve endothelial function.

Publication types

  • Comparative Study
  • Randomized Controlled Trial
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Atenolol / pharmacology*
  • Benzazepines / pharmacology*
  • Brachial Artery / drug effects
  • Brachial Artery / physiopathology
  • Cardiovascular Diseases / etiology
  • Cardiovascular Diseases / physiopathology
  • Cardiovascular Diseases / prevention & control*
  • Cyclic Nucleotide-Gated Cation Channels
  • Diabetes Mellitus, Type 2 / complications
  • Diabetes Mellitus, Type 2 / physiopathology*
  • Double-Blind Method
  • Electrocardiography
  • Endothelium, Vascular / drug effects*
  • Endothelium, Vascular / physiopathology
  • Female
  • Follow-Up Studies
  • Heart Rate / drug effects*
  • Humans
  • Ivabradine
  • Male
  • Middle Aged
  • Prospective Studies
  • Sympathetic Nervous System / drug effects
  • Sympatholytics / pharmacology
  • Vasodilation / drug effects

Substances

  • Benzazepines
  • Cyclic Nucleotide-Gated Cation Channels
  • Sympatholytics
  • Ivabradine
  • Atenolol