Pharmacotherapeutic considerations for the use of prasugrel and ticagrelor to reduce stent thrombosis in patients with acute coronary syndrome

Angiology. 2014 Feb;65(2):130-6. doi: 10.1177/0003319712467530. Epub 2012 Dec 4.

Abstract

Despite the improvement in stent technology, stent thrombosis (ST), a potentially catastrophic event, still occurs. Among several risk factors for ST, high on-treatment platelet reactivity to clopidogrel has been demonstrated to play a role, occurring in about one-third of the patients. In order to overcome this limitation, prasugrel and ticagrelor, newer P2Y12 inhibitors, have been developed and approved for clinical use. Two large clinical trials, TRial to assess Improvement in Therapeutic Outcomes by optimizing platelet inhibitioN with prasugrel-thrombolysis in myocardial infarction (TRITON-TIMI) 38 and Study of Platelet Inhibition and Patient Outcomes (PLATO), evaluated these drugs in patients with acute coronary syndrome (ACS), showing a significant improvement in efficacy end points (including a prominent reduction in ST occurrence) compared to clopidogrel. In contrast, the TRILOGY ACS trial found no benefit with prasugrel compared to clopidogrel in patients with medically treated ACS. The aim of this review is to consider decision-making strategies between prasugrel and ticagrelor in daily clinical practice.

Keywords: acute coronary syndromes; platelets; prasugrel; stent thrombosis; ticagrelor.

Publication types

  • Review

MeSH terms

  • Acute Coronary Syndrome
  • Adenosine / analogs & derivatives*
  • Adenosine / pharmacokinetics
  • Adenosine / pharmacology
  • Adenosine / therapeutic use
  • Coronary Thrombosis / prevention & control*
  • Humans
  • Myocardial Infarction / prevention & control
  • Percutaneous Coronary Intervention
  • Piperazines / pharmacokinetics
  • Piperazines / pharmacology
  • Piperazines / therapeutic use*
  • Platelet Aggregation Inhibitors / pharmacokinetics
  • Platelet Aggregation Inhibitors / pharmacology
  • Platelet Aggregation Inhibitors / therapeutic use*
  • Prasugrel Hydrochloride
  • Purinergic P2Y Receptor Antagonists / pharmacokinetics
  • Purinergic P2Y Receptor Antagonists / pharmacology
  • Purinergic P2Y Receptor Antagonists / therapeutic use*
  • Stents*
  • Thiophenes / pharmacokinetics
  • Thiophenes / pharmacology
  • Thiophenes / therapeutic use*
  • Ticagrelor

Substances

  • Piperazines
  • Platelet Aggregation Inhibitors
  • Purinergic P2Y Receptor Antagonists
  • Thiophenes
  • Prasugrel Hydrochloride
  • Ticagrelor
  • Adenosine