Cdk1 protein-mediated phosphorylation of receptor-associated protein 80 (RAP80) serine 677 modulates DNA damage-induced G2/M checkpoint and cell survival

J Biol Chem. 2013 Feb 8;288(6):3768-76. doi: 10.1074/jbc.M112.401299. Epub 2012 Dec 21.

Abstract

Post-translational phosphorylation plays critical roles in the assembly of signaling and repair proteins in the DNA damage response pathway. RAP80, a component of the BRCA1-A complex, is crucial in cell cycle checkpoint activation and DNA damage repair. However, its molecular mechanism is unclear. In this study, we identified Cdk1 as a new RAP80-binding protein and demonstrated that the Cdk1-cyclin B(1) complex phosphorylates RAP80 at Ser-677 using an in vitro kinase assay and a phosphopeptide-specific antibody against phospho-Ser-677 of RAP80. RAP80 Ser-677 phosphorylation occurred in the M phase of the cell cycle when Cdk1 was in an active state. In addition, ionizing radiation (IR) induced RAP80 phosphorylation at Ser-677. Mutation of Ser-677 to alanine sensitized cells to IR and functioned in G(2)/M checkpoint control. These results suggest that post-translational phosphorylation of RAP80 by the Cdk1-cyclin B(1) complex is important for RAP80 functional sensitivity to IR and G(2)/M checkpoint control.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Substitution
  • CDC2 Protein Kinase / genetics
  • CDC2 Protein Kinase / metabolism*
  • Carrier Proteins / genetics
  • Carrier Proteins / metabolism*
  • Cell Survival / genetics
  • Cyclin B1 / genetics
  • Cyclin B1 / metabolism
  • DNA Damage*
  • DNA-Binding Proteins
  • G2 Phase Cell Cycle Checkpoints*
  • HeLa Cells
  • Histone Chaperones
  • Humans
  • M Phase Cell Cycle Checkpoints*
  • Mutation, Missense
  • Nuclear Proteins / genetics
  • Nuclear Proteins / metabolism*
  • Phosphorylation / genetics
  • Protein Processing, Post-Translational*
  • Serine

Substances

  • CCNB1 protein, human
  • Carrier Proteins
  • Cyclin B1
  • DNA-Binding Proteins
  • Histone Chaperones
  • Nuclear Proteins
  • UIMC1 protein, human
  • Serine
  • CDC2 Protein Kinase