In vivo effects of recombinant human interleukin-6 in primates: stimulated production of platelets

Blood. 1990 Apr 15;75(8):1602-5.

Abstract

In cynomolgus monkeys, twice daily subcutaneous injections of recombinant human interleukin-6 (rhIL-6) at doses of 5 to 80 micrograms/kg/d for 14 consecutive days caused dose-dependent increases in platelet count, usually continuing for more than 1 week after cessation of the injections. The count reached a level approximately twofold or more above the preinjection level even at 5 micrograms/kg/d, and at doses of more than 20 micrograms/kg/d, the increase became biphasic with a higher second peak 3 days after cessation of the injections. Morphologic analysis of the bone marrow after the 7 day-injections with 80 micrograms/kg/d revealed a marked increment in size of megakaryocytes compared with control, indicating the promotion of megakaryocyte maturation. Other changes attributable to the rhIL-6 treatment include dose-dependent loss of body weight, anemia, neutrophilia and monocytosis, elevation of serum C-reactive protein and alpha-1 acid glycoprotein levels, and decrease of serum albumin; all of which returned to normal within 1 week after cessation of the injections and were tolerable at doses of less than 10 micrograms/kg/d. These findings suggest that rhIL-6 may be an effective strategy for the treatment of thrombocytopenia.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Blood Cell Count / drug effects
  • Blood Platelets / cytology
  • Blood Platelets / drug effects*
  • Body Weight / drug effects
  • Bone Marrow / drug effects
  • Bone Marrow Cells
  • Cell Division / drug effects
  • Dose-Response Relationship, Drug
  • Female
  • Injections
  • Interleukin-6 / administration & dosage
  • Interleukin-6 / pharmacology*
  • Interleukin-6 / physiology
  • Macaca / blood*
  • Macaca fascicularis / blood*
  • Megakaryocytes / drug effects
  • Recombinant Proteins / pharmacology*
  • Recombinant Proteins / physiology

Substances

  • Interleukin-6
  • Recombinant Proteins