Efficacy and safety of long acting injectable atypical antipsychotics: a review

Curr Clin Pharmacol. 2013 Aug;8(3):256-64. doi: 10.2174/15748847113089990056.

Abstract

Schizophrenia is a chronic, severe and recurrent brain disorder that requires continuous, long-term treatment with antipsychotic medication to minimize relapse and provide clinical benefit to patients. For patients with schizophrenia, non-adherence to medication is a major risk factor for relapse and re-hospitalization. Long-acting injectable formulations of second-generation antipsychotics (SGAs-LAIs) provide constant medication delivery and the potential for improved adherence. Currently, three drugs are available for the treatment of schizophrenia, risperidone longacting injectable, olanzapine pamoate and paliperidone palmitate. Several studies have also demonstrated efficacy and safety of such drugs in patients with acute schizophrenia. In the present paper the literature on LAI atypical antipsychotics will be reviewed and practical advice will be given concerning the use of these drugs in the clinical practice.

Publication types

  • Review

MeSH terms

  • Antipsychotic Agents / administration & dosage
  • Antipsychotic Agents / adverse effects
  • Antipsychotic Agents / therapeutic use*
  • Benzodiazepines / administration & dosage
  • Benzodiazepines / adverse effects
  • Benzodiazepines / therapeutic use
  • Delayed-Action Preparations
  • Drug Delivery Systems*
  • Humans
  • Injections
  • Isoxazoles / administration & dosage
  • Isoxazoles / adverse effects
  • Isoxazoles / therapeutic use
  • Medication Adherence
  • Olanzapine
  • Paliperidone Palmitate
  • Palmitates / administration & dosage
  • Palmitates / adverse effects
  • Palmitates / therapeutic use
  • Risperidone / administration & dosage
  • Risperidone / adverse effects
  • Risperidone / therapeutic use
  • Schizophrenia / drug therapy*
  • Schizophrenia / physiopathology

Substances

  • Antipsychotic Agents
  • Delayed-Action Preparations
  • Isoxazoles
  • Palmitates
  • Benzodiazepines
  • Risperidone
  • Olanzapine
  • Paliperidone Palmitate