[Effect of tetramethylpyrazine on Nogo gene regulation of the proliferation in cardiac fibroblast]

Sichuan Da Xue Xue Bao Yi Xue Ban. 2012 Nov;43(6):843-6.
[Article in Chinese]

Abstract

Objective: To investigate the effects of different doses of Tetramethylpyrazine (TMP) on collagen synthesis and Nogo expression in cardiac fibroblasts and the potential role of Nogo in myocardial fibrosis.

Methods: The cultured neonatal rat cardiac fibroblasts were induced by angiotensin II and TMP at the same time. The mRNA expression of Nogo-A, Nogo-B and collagen I were detected with real-time fluorescence quantitative PCR. And Nogo protein was semi-quantitatively detected by using Western blot method.

Results: Under the intervention of TMP, the increased mRNA expression of Nogo-A and collagen I induced by angiotensin II were decreased, while the decreased mRNA expression of Nogo-B was increased. Compared with the control group, the expression of Nogo-A protein and Nogo-B protein showed similar changes as evaluated with Western blot.

Conclusion: TMP could inhibit collagen synthesis in cardiac fibroblast induced by angiotensin II. The accompanying differential expression of Nogo-A and Nogo-B indicated that the anti-fibrosis effect of TMP might be related to the regulation effects of Nogo gene.

MeSH terms

  • Angiotensin II / pharmacology
  • Animals
  • Animals, Newborn
  • Cell Proliferation / drug effects*
  • Cells, Cultured
  • Collagen Type I / metabolism
  • Fibroblasts / cytology
  • Fibroblasts / drug effects*
  • Gene Expression Regulation
  • Male
  • Myelin Proteins / genetics
  • Myelin Proteins / metabolism*
  • Myocytes, Cardiac / cytology
  • Myocytes, Cardiac / drug effects*
  • Nogo Proteins
  • Pyrazines / pharmacology*
  • RNA, Messenger / genetics
  • RNA, Messenger / metabolism
  • Rats
  • Rats, Sprague-Dawley

Substances

  • Collagen Type I
  • Myelin Proteins
  • Nogo Proteins
  • Pyrazines
  • RNA, Messenger
  • Rtn4 protein, rat
  • Angiotensin II
  • tetramethylpyrazine