Erythrocyte membrane-cloaked polymeric nanoparticles for controlled drug loading and release

Nanomedicine (Lond). 2013 Aug;8(8):1271-80. doi: 10.2217/nnm.12.153. Epub 2013 Feb 14.

Abstract

Aim: Polymeric nanoparticles (NPs) cloaked by red blood cell membrane (RBCm) confer the combined advantage of both long circulation lifetime and controlled drug release. The authors carried out studies to gain a better understanding of the drug loading, drug-release kinetics and cell-based efficacy of RBCm-cloaked NPs.

Materials & methods: Two strategies for loading doxorubicin into the RBCm-cloaked NPs were compared: physical encapsulation and chemical conjugation. In vitro efficacy was examined using the acute myeloid leukemia cell line, Kasumi-1.

Results: It was found that the chemical conjugation strategy resulted in a more sustained drug release profile, and that the RBCm cloak provided a barrier, retarding the outward diffusion of encapsulated drug molecules. It was also demonstrated that RBCm-cloaked NPs exhibit higher toxicity in comparison with free doxorubicin.

Conclusion: These results indicate that the RBCm-cloaked NPs hold great promise to become a valuable drug-delivery platform for the treatment of various diseases such as blood cancers.

Publication types

  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Cell Line, Tumor
  • Cell Survival / drug effects*
  • Delayed-Action Preparations / chemistry
  • Doxorubicin / administration & dosage
  • Doxorubicin / chemistry
  • Drug Delivery Systems
  • Erythrocyte Membrane / chemistry*
  • Humans
  • Leukemia, Myeloid, Acute / drug therapy*
  • Leukemia, Myeloid, Acute / pathology
  • Nanoparticles / administration & dosage*
  • Nanoparticles / chemistry
  • Polymers / administration & dosage
  • Polymers / chemistry

Substances

  • Delayed-Action Preparations
  • Polymers
  • Doxorubicin