Effect of rice cell-derived human granulocyte-macrophage colony-stimulating factor on 5-fluorouracil-induced mucositis in hamsters

Biol Pharm Bull. 2013;36(3):425-31. doi: 10.1248/bpb.b12-00869.

Abstract

Granulocyte-macrophage colony-stimulating factor (GM-CSF) is an important regulator of the maturation and function of cells in the granulocyte and macrophage lineages, and also plays a significant role in wound healing. In a previous study, we expressed human GM-CSF in rice cells (rice cell-derived human GM-CSF; rhGM-CSF). The purpose of the present study was to evaluate its effect on wound healing in oral mucositis. Oral mucositis was induced in Syrian hamster cheek pouches by 5-fluorouracil treatment and mechanical scratching. Ulcerated areas were treated from days 3 to 14 with an application of 200 µL saline, or of the same volume of a solution containing 0.04, 0.2, or 1 µg/mL rhGM-CSF. Treatment of hamsters with rhGM-CSF reduced the ulcerated areas of the oral mucosa, compared with the control. Early in the healing process, the mucositis tissue layer of the rhGM-CSF-treated group showed significantly decreased myeloperoxidase activity and increased numbers of proliferating cell nuclear antigen (PCNA)-positive cells. Treatment with rhGM-CSF also affected expression of inflammatory cytokines in the ulcerative mucosal tissue. These results demonstrate the efficacy of plant-produced rhGM-CSF in wound healing and have significant implications for the development of rhGM-CSF as a therapeutic agent for ulcerative oral mucositis.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Antimetabolites, Antineoplastic / toxicity*
  • Cricetinae
  • Fluorouracil / toxicity*
  • Granulocyte-Macrophage Colony-Stimulating Factor / therapeutic use*
  • Interleukin-1beta / genetics
  • Male
  • Mesocricetus
  • Mouth Mucosa / drug effects
  • Mouth Mucosa / enzymology
  • Oryza / genetics
  • Peroxidase / metabolism
  • Proliferating Cell Nuclear Antigen / analysis
  • Recombinant Proteins / therapeutic use
  • Stomatitis / chemically induced
  • Stomatitis / drug therapy*
  • Stomatitis / pathology
  • Transforming Growth Factor beta / genetics
  • Wound Healing / drug effects

Substances

  • Antimetabolites, Antineoplastic
  • Interleukin-1beta
  • Proliferating Cell Nuclear Antigen
  • Recombinant Proteins
  • Transforming Growth Factor beta
  • Granulocyte-Macrophage Colony-Stimulating Factor
  • Peroxidase
  • Fluorouracil