Polymerization of a peptide-based enzyme substrate

Chem Commun (Camb). 2013 Apr 11;49(28):2873-5. doi: 10.1039/c3cc40472b.

Abstract

Polymers of norbornenyl-modified peptide-based enzyme substrates have been prepared via ring-opening metathesis polymerization (ROMP). Peptides displayed on water-soluble homopolymers retain the ability to be enzymatically processed by a disease-associated enzyme. In contrast, when the peptides are densely arrayed on a nanoparticle derived from a self-assembled amphiphilic block-copolymer, they function with reduced activity as enzymatic substrates.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Enzymes / metabolism*
  • Humans
  • Nanoparticles / chemistry
  • Oligopeptides / chemistry*
  • Oligopeptides / metabolism*
  • Polymerization*
  • Proteolysis

Substances

  • Enzymes
  • Oligopeptides