Tumor-suppressive maspin functions as a reactive oxygen species scavenger: importance of cysteine residues

J Biol Chem. 2013 Apr 19;288(16):11611-20. doi: 10.1074/jbc.M112.410852. Epub 2013 Mar 7.

Abstract

Maspin is a member of the serine protease inhibitor (serpin) superfamily and displays tumor-suppressing activity by controlling cell migration, proliferation, apoptosis, and adhesion. Here, we provide evidence that maspin acts as a reactive oxygen species (ROS) scavenger through oxidation of three structurally exposed cysteine thiols to sulfenic acid. Ablation of these cysteine residues in maspin resulted in a significant increase in total ROS production in mouse mammary TM40D cells. Also, cells containing a triple-cysteine mutant of maspin showed elevated ERK1/2 activity, a downstream target of ROS, and enhanced proliferation and colony formation. These findings establish a novel mechanism by which maspin utilizes its cysteine thiols to inhibit oxidative stress and cell growth.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Amino Acid Substitution
  • Animals
  • Cell Line, Tumor
  • Cell Proliferation
  • Cysteine / genetics
  • Cysteine / metabolism*
  • Female
  • Free Radical Scavengers / metabolism*
  • MAP Kinase Signaling System / genetics
  • Mice
  • Mutation, Missense
  • Oxidation-Reduction
  • Oxidative Stress*
  • Reactive Oxygen Species / metabolism*
  • Serpins / genetics
  • Serpins / metabolism*
  • Tumor Suppressor Proteins / genetics
  • Tumor Suppressor Proteins / metabolism*

Substances

  • Free Radical Scavengers
  • Reactive Oxygen Species
  • SERPIN-B5
  • Serpins
  • Tumor Suppressor Proteins
  • Cysteine