Cocaine-induced reduction of glucose utilization in human brain. A study using positron emission tomography and [fluorine 18]-fluorodeoxyglucose

Arch Gen Psychiatry. 1990 Jun;47(6):567-74. doi: 10.1001/archpsyc.1990.01810180067010.

Abstract

We examined the effects of cocaine hydrochloride (40 mg intravenously) on regional cerebral metabolic rates for glucose and on subjective self-reports of eight polydrug abusers in a double-blind, placebo-controlled, crossover study. The regional cerebral metabolic rate for glucose was measured by the [fluorine 18]-fluorodeoxyglucose method, using positron emission tomography. With eyes covered, subjects listened to a tape that presented white noise, "beep" prompts, and questions about subjective effects of cocaine or saline. Cocaine produced euphoria and reduced glucose utilization globally (mean reduction, 14%). Twenty-six of 29 brain regions (all neocortical areas, basal ganglia, portions of the hippocampal formation, thalamus, and midbrain) showed significant decrements (5% to 26%) in the regional cerebral metabolic rate for glucose. No significant effects of cocaine were observed in the pons, the cerebellar cortex, or the vermis. Right-greater-than-left hemispheric asymmetry of regional cerebral metabolic rates for glucose occurred in the lateral thalamus. The findings demonstrate that reduced cerebral metabolism is associated with cocaine-induced euphoria.

Publication types

  • Clinical Trial
  • Controlled Clinical Trial
  • Randomized Controlled Trial
  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Adult
  • Blood Pressure / drug effects
  • Brain / drug effects
  • Brain / metabolism*
  • Cerebral Cortex / drug effects
  • Cerebral Cortex / metabolism
  • Cocaine / pharmacology*
  • Deoxyglucose / analogs & derivatives
  • Deoxyglucose / metabolism
  • Double-Blind Method
  • Euphoria
  • Fluorodeoxyglucose F18
  • Glucose / metabolism*
  • Heart Rate / drug effects
  • Humans
  • Male
  • Placebos
  • Substance-Related Disorders* / metabolism
  • Substance-Related Disorders* / psychology
  • Tomography, Emission-Computed

Substances

  • Placebos
  • Fluorodeoxyglucose F18
  • Deoxyglucose
  • Cocaine
  • Glucose