Stimulation of A2B adenosine receptors protects against trauma-hemorrhagic shock-induced lung injury

Purinergic Signal. 2013 Sep;9(3):427-32. doi: 10.1007/s11302-013-9362-7. Epub 2013 Apr 13.

Abstract

Inflammation is responsible for secondary organ failure after trauma and hemorrhagic shock (T/HS). Adenosine, acting through four G protein-coupled cell surface receptors, A1, A2A, A2B, and A3, exerts a number of tissue protective and anti-inflammatory effects. The goal of the present study was to test the effect of A2B adenosine receptor stimulation on T/HS-induced organ injury and inflammation in rats. Rats after T/HS were resuscitated with Ringer's lactate containing the A2B receptor agonist BAY 60-6583 or its vehicle. We found that BAY 60-6583 decreased T/HS-induced lung permeability and plasma creatine kinase levels but failed to affect T/HS-induced lung neutrophil infiltration and IκBα expression and plasma alanine aminotransferase levels. Thus, we conclude that stimulation of A2B receptors protects against T/HS-induced lung and muscle injury.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Acute Lung Injury / metabolism*
  • Aminopyridines / pharmacology
  • Animals
  • Blotting, Western
  • Disease Models, Animal
  • Inflammation / metabolism*
  • Male
  • Purinergic P1 Receptor Agonists / pharmacology
  • Rats
  • Rats, Sprague-Dawley
  • Receptor, Adenosine A2B / metabolism*
  • Shock, Hemorrhagic / metabolism*
  • Wounds and Injuries

Substances

  • Aminopyridines
  • BAY 60-6583
  • Purinergic P1 Receptor Agonists
  • Receptor, Adenosine A2B