Targeting deregulated epigenetic control in cancer

J Cell Physiol. 2013 Nov;228(11):2103-8. doi: 10.1002/jcp.24387.

Abstract

Cancer is a multifaceted disease that involves acquisition of genetic mutations, deletions, and amplifications as well as deregulation of epigenetic mechanisms that fine-tune gene regulation. Key epigenetic mechanisms that include histone modifications, DNA methylation, and non-coding RNA-mediated gene silencing are often deregulated in a variety of cancers. Subnuclear localization of key proteins in the interphase nucleus and bookmarking of genes by lineage commitment factors in mitosis-a new dimension to epigenetic control of fundamental biological processes-is also modified in cancer. In this review, we discuss the various aspects of epigenetic control that are operative in a variety of cancers and their potential for risk assessment, early detection, targeted therapy, and personalized medicine.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't
  • Review

MeSH terms

  • Animals
  • DNA Methylation / genetics
  • Epigenesis, Genetic*
  • Histones / metabolism
  • Humans
  • Neoplasms / genetics*
  • RNA, Untranslated / metabolism
  • Translational Research, Biomedical

Substances

  • Histones
  • RNA, Untranslated