Targeting inflammasomes in rheumatic diseases

Nat Rev Rheumatol. 2013 Jul;9(7):391-9. doi: 10.1038/nrrheum.2013.61. Epub 2013 May 14.

Abstract

Inflammasomes are key inducers of inflammation in response to exogenous and endogenous stimuli, because they regulate the processing and secretion of the proinflammatory cytokines IL-1β and IL-18. Thus, inflammasomes have a crucial role in host defence against infection, but they can also be involved in inflammatory diseases. Indeed, the NLRP3 (NOD-, LRR- and pyrin domain-containing 3) inflammasome has been shown to play a part in several inflammatory rheumatic disorders, although the mechanisms involved are better elucidated in some of these diseases than in others. In particular, the pathogenesis of cryopyrin-associated periodic syndromes and microcrystal-induced arthritides is thought to be dependent on activation of the NLRP3 inflammasome, and IL-1 inhibition has shown efficacy as a therapeutic strategy in both groups of conditions. In this Review, we describe the current understanding of the mechanisms that trigger the inflammasome, and consider the relevance of the inflammasome to a variety of rheumatic diseases. In addition, we discuss the current therapies targeting this molecular complex, as well as future therapeutic prospects.

Publication types

  • Research Support, Non-U.S. Gov't
  • Review

MeSH terms

  • Carrier Proteins / physiology
  • Cryopyrin-Associated Periodic Syndromes / drug therapy
  • Cryopyrin-Associated Periodic Syndromes / physiopathology
  • Humans
  • Inflammasomes / physiology*
  • Interleukin-1 / physiology
  • Interleukin-18 / physiology
  • NLR Family, Pyrin Domain-Containing 3 Protein
  • Rheumatic Diseases / drug therapy*
  • Rheumatic Diseases / physiopathology*

Substances

  • Carrier Proteins
  • Inflammasomes
  • Interleukin-1
  • Interleukin-18
  • NLR Family, Pyrin Domain-Containing 3 Protein
  • NLRP3 protein, human