Apolipoproteins E and AV mediate lipoprotein clearance by hepatic proteoglycans

J Clin Invest. 2013 Jun;123(6):2742-51. doi: 10.1172/JCI67398. Epub 2013 May 8.

Abstract

The heparan sulfate proteoglycan (HSPG) syndecan-1 (SDC1) acts as a major receptor for triglyceride-rich lipoprotein (TRL) clearance in the liver. We sought to identify the relevant apolipoproteins on TRLs that mediate binding to SDC1 and determine their clinical relevance. Evidence supporting ApoE as a major determinant arose from its enrichment in TRLs from mice defective in hepatic heparan sulfate (Ndst1f/fAlbCre⁺ mice), decreased binding of ApoE-deficient TRLs to HSPGs on human hepatoma cells, and decreased clearance of ApoE-deficient [³H]TRLs in vivo. Evidence for a second ligand was suggested by the faster clearance of ApoE-deficient TRLs after injection into WT Ndst1f/fAlbCre⁻ versus mutant Ndst1f/fAlbCre⁺ mice and elevated fasting and postprandial plasma triglycerides in compound Apoe⁻/⁻Ndst1f/fAlbCre⁺ mice compared with either single mutant. ApoAV emerged as a candidate based on 6-fold enrichment of ApoAV in TRLs accumulating in Ndst1f/fAlbCre⁺ mice, decreased binding of TRLs to proteoglycans after depletion of ApoAV or addition of anti-ApoAV mAb, and decreased heparan sulfate-dependent binding of ApoAV-deficient particles to hepatocytes. Importantly, disruption of hepatic heparan sulfate-mediated clearance increased atherosclerosis. We conclude that clearance of TRLs by hepatic HSPGs is atheroprotective and mediated by multivalent binding to ApoE and ApoAV.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Aorta, Thoracic / metabolism
  • Aorta, Thoracic / pathology
  • Apolipoprotein A-V
  • Apolipoproteins / metabolism*
  • Apolipoproteins B / metabolism
  • Apolipoproteins E / metabolism*
  • Atherosclerosis / blood
  • Atherosclerosis / pathology
  • Cell Line, Tumor
  • Female
  • Humans
  • Lipoproteins / metabolism
  • Liver / metabolism
  • Male
  • Mice
  • Mice, Transgenic
  • Protein Binding
  • Syndecan-1 / metabolism*
  • Triglycerides / blood

Substances

  • Apoa5 protein, mouse
  • Apolipoprotein A-V
  • Apolipoproteins
  • Apolipoproteins B
  • Apolipoproteins E
  • Lipoproteins
  • Sdc1 protein, mouse
  • Syndecan-1
  • Triglycerides