Development of acneiform rash does not predict response to lapatinib treatment in patients with breast cancer

Pharmacotherapy. 2013 Oct;33(10):1126-9. doi: 10.1002/phar.1308. Epub 2013 Jun 6.

Abstract

Study objective: To determine if development of acneiform rash is a predictor of objective response rate with lapatinib.

Design: Subanalysis of data from a prospective, phase II study.

Setting: Academic breast care clinic.

Patients: Forty-nine treatment-naïve patients with human epidermal growth factor receptor-2 (HER2)-positive locally advanced breast cancer, who were treated with neoadjuvant lapatinib monotherapy for 6 weeks; 47 patients were included in the final analysis.

Measurements and main results: Of the 49 patients enrolled, 33 (67%) developed a rash of any type, and 26 (55%) had acneiform rash. Of the 26 evaluable patients with acneiform rash (55%), 19 (73%) responded to lapatinib and 7 (27%) did not. Of the 21 evaluable patients without acneiform rash, 11 (67%) responded to treatment and 7 (33%) did not. Thus, no association was found between the occurrence of acneiform rash and response to lapatinib monotherapy.

Conclusion: This study does not support the development of the acneiform rash as a predictor of clinical efficacy of lapatinib in the treatment of breast cancer.

Keywords: EGFR; HER2; breast cancer; dermatologic toxicity; lapatinib; rash.

Publication types

  • Clinical Trial, Phase II

MeSH terms

  • Acneiform Eruptions / chemically induced*
  • Acneiform Eruptions / pathology
  • Adult
  • Aged
  • Aged, 80 and over
  • Antineoplastic Agents / adverse effects
  • Antineoplastic Agents / therapeutic use*
  • Breast Neoplasms / drug therapy
  • Breast Neoplasms / pathology
  • Drug Eruptions / etiology*
  • Drug Eruptions / pathology
  • Female
  • Humans
  • Lapatinib
  • Middle Aged
  • Neoadjuvant Therapy
  • Prospective Studies
  • Quinazolines / adverse effects
  • Quinazolines / therapeutic use*
  • Receptor, ErbB-2 / metabolism
  • Treatment Outcome

Substances

  • Antineoplastic Agents
  • Quinazolines
  • Lapatinib
  • ERBB2 protein, human
  • Receptor, ErbB-2