Thymol from Thymus quinquecostatus Celak. protects against tert-butyl hydroperoxide-induced oxidative stress in Chang cells

J Nat Med. 2014 Jan;68(1):154-62. doi: 10.1007/s11418-013-0786-8. Epub 2013 Jun 15.

Abstract

The present work describes the protective effects of thymol isolated from Thymus quinquecostatus Celak. against tert-butyl hydroperoxide (t-BHP)-induced oxidative damage through various experiments with Chang liver cells. Thymol significantly protected hepatocytes against t-BHP-induced cell cytotoxicity as demonstrated by increased viability. Furthermore, observation of Hoechst staining, annexin V/PI staining, and expression of Bcl-2 and Bax indicated that thymol inhibited t-BHP-induced Chang cell damage. Further, thymol inhibited the loss of mitochondrial membrane potential in t-BHP-treated Chang cells and prevented oxidative stress-triggered reactive oxygen species (ROS) and lipid peroxidation (malondialdehyde, MDA). Thymol restored the antioxidant capability of hepatocytes including glutathione (GSH) levels which were reduced by t-BHP. These results indicated that thymol prevents oxidative stress-induced damage to liver cells through suppression of ROS and MDA levels and increase of GSH level.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Annexin A5 / metabolism
  • Antioxidants / isolation & purification
  • Antioxidants / pharmacology*
  • Apoptosis / drug effects
  • Cell Survival / drug effects
  • Cytoprotection
  • Dose-Response Relationship, Drug
  • Glutathione / metabolism
  • Glutathione / pharmacology
  • Hepatocytes / drug effects*
  • Hepatocytes / metabolism
  • Hepatocytes / pathology
  • Humans
  • Lipid Peroxidation / drug effects
  • Malondialdehyde / metabolism
  • Membrane Potential, Mitochondrial / drug effects
  • Oxidative Stress / drug effects*
  • Phytotherapy
  • Plants, Medicinal
  • Reactive Oxygen Species / metabolism
  • Thymol / isolation & purification
  • Thymol / pharmacology*
  • Thymus Plant* / chemistry
  • bcl-2-Associated X Protein / metabolism
  • tert-Butylhydroperoxide / toxicity*

Substances

  • Annexin A5
  • Antioxidants
  • BAX protein, human
  • Reactive Oxygen Species
  • bcl-2-Associated X Protein
  • Thymol
  • Malondialdehyde
  • tert-Butylhydroperoxide
  • Glutathione